DK138496B - Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.

Info

Publication number
DK138496B
DK138496B DK34572AA DK34572A DK138496B DK 138496 B DK138496 B DK 138496B DK 34572A A DK34572A A DK 34572AA DK 34572 A DK34572 A DK 34572A DK 138496 B DK138496 B DK 138496B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
imidazoline derivatives
analogous process
Prior art date
Application number
DK34572AA
Other languages
English (en)
Other versions
DK138496C (da
Inventor
Fernand Binon
Alex Areschka
Original Assignee
Labaz
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Labaz filed Critical Labaz
Publication of DK138496B publication Critical patent/DK138496B/da
Application granted granted Critical
Publication of DK138496C publication Critical patent/DK138496C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK34572AA 1971-01-27 1972-01-26 Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. DK138496B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB332771 1971-01-27

Publications (2)

Publication Number Publication Date
DK138496B true DK138496B (da) 1978-09-18
DK138496C DK138496C (da) 1979-02-26

Family

ID=9756227

Family Applications (1)

Application Number Title Priority Date Filing Date
DK34572AA DK138496B (da) 1971-01-27 1972-01-26 Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.

Country Status (17)

Country Link
US (1) US3818035A (da)
JP (1) JPS4938273B1 (da)
AT (1) AT311336B (da)
BE (1) BE777689A (da)
CA (1) CA962273A (da)
CH (1) CH535254A (da)
DE (1) DE2203373C3 (da)
DK (1) DK138496B (da)
FI (1) FI55841C (da)
GB (1) GB1333471A (da)
HU (1) HU162823B (da)
NL (1) NL150454B (da)
NO (1) NO134115C (da)
SE (1) SE378426B (da)
SU (1) SU474145A3 (da)
YU (1) YU34694B (da)
ZA (1) ZA72286B (da)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3927023A (en) * 1974-05-24 1975-12-16 Warner Lambert Co Imidazolyl benzofurans
DE3049542A1 (de) * 1980-12-31 1982-07-29 Basf Ag, 6700 Ludwigshafen Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung
ZA825413B (en) * 1981-08-26 1983-06-29 Pfizer Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them
US4806663A (en) * 1987-04-06 1989-02-21 The University Of Tennessee Research Corporation Certain 3-substituted 2-alkyl benzofuran derivatives
US4851554A (en) * 1987-04-06 1989-07-25 University Of Tennessee Research Corporation Certain 3-substituted 2-alkyl benzofuran derivatives
US4831156A (en) * 1987-09-30 1989-05-16 The University Of Tennessee Research Corp. 3-substituted 2-alkyl indole derivatives
WO1999032482A1 (en) * 1997-12-19 1999-07-01 Eli Lilly And Company Hypoglycemic imidazoline compounds
US7777035B2 (en) * 2005-06-22 2010-08-17 Chemocentryx, Inc. Azaindazole compounds and methods of use
KR20080080410A (ko) * 2006-01-27 2008-09-03 에프. 호프만-라 로슈 아게 이미다졸린 유도체의 치환된 2-이미다졸의 용도
CA2665255A1 (en) * 2006-10-19 2008-04-24 F. Hoffmann-La Roche Ag Aminomethyl-2-imidazoles with affinity with the trace amine associated receptors
BRPI0717939A2 (pt) * 2006-10-19 2013-12-03 Hoffmann La Roche Aminometil-4-imidazóis
BRPI0718054A2 (pt) * 2006-11-02 2013-11-05 Hoffmann La Roche 2-imidazóis substituídos como moduladores de receptores associados à traços de aminas
JP2010510184A (ja) * 2006-11-16 2010-04-02 エフ．ホフマン−ラ ロシュ アーゲー 置換４−イミダゾール類
BRPI0720047A2 (pt) * 2006-12-13 2013-12-24 Hoffmann La Roche 2-imidazóis como ligantes para receptores associados a aminas de traço (taar)
US20080146523A1 (en) * 2006-12-18 2008-06-19 Guido Galley Imidazole derivatives
RU2473545C2 (ru) * 2007-02-02 2013-01-27 Ф.Хоффманн-Ля Рош Аг Новые 2-аминооксазолины в качестве лигандов taar1 для заболеваний цнс
KR101222412B1 (ko) * 2007-02-15 2013-01-15 에프. 호프만-라 로슈 아게 Ｔａａｒ1 리간드로서의 2-아미노옥사졸린
CA2691082A1 (en) 2007-07-02 2009-01-08 F. Hoffmann-La Roche Ag 2 -imidazolines having a good affinity to the trace amine associated receptors (taars)
WO2009003867A1 (en) * 2007-07-03 2009-01-08 F. Hoffmann-La Roche Ag 4-imidazolines and their use as antidepressants
AU2008281918A1 (en) * 2007-07-27 2009-02-05 F. Hoffmann-La Roche Ag 2-azetidinemethaneamines and 2-pyrrolidinemethaneamines as TAAR-ligands
JP2010535172A (ja) * 2007-08-02 2010-11-18 エフ．ホフマン−ラ ロシュ アーゲー Ｃｎｓ障害の処置のためのベンズアミド誘導体の使用
CA2695331A1 (en) * 2007-08-03 2009-02-12 F. Hoffmann-La Roche Ag Pyridinecarboxamide and benzamide derivatives as taar1 ligands
US8242153B2 (en) * 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
JP5547187B2 (ja) * 2008-07-24 2014-07-09 エフ．ホフマン−ラ ロシュ アーゲー ４，５−ジヒドロ−オキサゾール−２−イル誘導体
US20100311798A1 (en) * 2009-06-05 2010-12-09 Decoret Guillaume 2-aminooxazolines as taar1 ligands
US8354441B2 (en) * 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
SG11201807516UA (en) 2016-03-17 2018-09-27 Hoffmann La Roche 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1121054B (de) * 1960-11-23 1962-01-04 Merck Ag E Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen

Also Published As

Publication number Publication date
NL150454B (nl) 1976-08-16
NO134115B (da) 1976-05-10
AT311336B (de) 1973-11-12
FI55841B (fi) 1979-06-29
NL7201121A (da) 1972-07-31
YU34694B (en) 1979-12-31
HU162823B (da) 1973-04-28
AU3817772A (en) 1973-07-26
DE2203373B2 (de) 1977-08-11
CH535254A (fr) 1973-03-31
ZA72286B (en) 1972-09-27
GB1333471A (en) 1973-10-10
US3818035A (en) 1974-06-18
SU474145A3 (ru) 1975-06-14
DE2203373C3 (de) 1978-04-13
BE777689A (fr) 1972-07-05
CA962273A (en) 1975-02-04
DK138496C (da) 1979-02-26
NO134115C (da) 1976-08-18
DE2203373A1 (de) 1972-08-17
SE378426B (da) 1975-09-01
JPS4938273B1 (da) 1974-10-16
FI55841C (fi) 1979-10-10
YU18172A (en) 1979-07-10

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