KEGG   DGROUP: Bosentan
Entry
DG00266                     DGroup                                 
Name
Bosentan
Type
Chemical
Member
D07538  
Bosentan (INN)
D01227  
Bosentan (USAN); Bosentan hydrate (JAN)  <JP/US>
Class
Cardiovascular agent
 DG01502  Endothelin receptor antagonist
Metabolizing enzyme substrate
 DG01642  CYP2C9 substrate
 DG01633  CYP3A/CYP3A4 substrate
  DG02913  CYP3A4 substrate
Metabolizing enzyme inducer
 DG02886  CYP2C9 inducer
 DG02853  CYP3A/CYP3A4 inducer
  DG01635  CYP3A4 inducer
Remark
ATC code: C02KX01
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