| Esterified local anesthetic |
| Metabutethamine |
| Procaine |
| Procaine (INN) |
| Procaine hydrochloride (JP18/USP) <JP> |
| Tetracaine |
| Tetracaine (USP/INN) |
| Tetracaine hydrochloride (JP18/USP) <US> |
| Chloroprocaine |
| Chloroprocaine (INN) |
| Chloroprocaine hydrochloride (USP) <US> |
| Cocaine |
| Cocaine (USP) |
| Cocaine hydrochloride (JP18/USP) <US> |
| Aminobenzoic acid |
| Aminobenzoic acid (USP) |
| Benzocaine (USP/INN); Ethyl aminobenzoate (JP18) <JP> |
| Aminobenzoate potassium (USP) |
| Aminobenzoate sodium (USP) |
| Amide type local anesthetic |
| Bupivacaine |
| Bupivacaine (USAN/INN) <US> |
| Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18) <JP/US> |
| Lidocaine |
| Lidocaine (JP18/USP/INN) <JP/US> |
| Lidocaine hydrochloride (JAN/USP) <JP/US> |
| Lidocaine hydrochloride monohydrate <JP/US> |
| Mepivacaine |
| Mepivacaine (INN) |
| Mepivacaine hydrochloride (JP18/USP) <JP/US> |
| Prilocaine |
| Prilocaine (USP/INN); Propitocaine (JAN) |
| Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN) <US> |
| Butanilicaine (INN) |
| Dibucaine |
| Dibucaine (USP); Cinchocaine (INN) |
| Dibucaine hydrochloride (JP18/USP) |
| Etidocaine |
| Etidocaine (USAN/INN) |
| Etidocaine hydrochloride |
| Articaine |
| Articaine (INN) |
| Articaine hydrochloride (JAN/USP) |
| Ropivacaine |
| Ropivacaine (INN) |
| Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN) <JP/US> |
| Levobupivacaine |
| Levobupivacaine (INN) |
| Levobupivacaine hydrochloride (JAN/USAN) <JP> |
| Oxetacaine |
| Oxethazaine (JP18/USAN); Oxetacaine (INN) <JP> |
| Oxetacaine hydrochloride |
| Trimecaine |
| Trimecaine (INN) |
| Trimecaine hydrochloride |
| Tolycaine hydrochloride (JAN) |
| Dexivacaine (USAN/INN) |
| Pyrrocaine (USAN/INN) |
| Rodocaine (USAN) |
| Ethyl chloride (USP) |
| Dyclonine |
| Dyclonine (INN) |
| Dyclonine hydrochloride (USP) <US> |
| Phenol |
| Phenol (JP18/USP); Liquefied phenol (JP18); Phenol for disinfection (JP18) <JP> |
| Phenolated water (JP18); Phenolated water for disinfection (JP18) <JP> |
| Capsaicin (JAN/USP) <US> |
| Oxybuprocaine |
| Oxybuprocaine (INN) |
| Benoxinate hydrochloride (USP); Oxybuprocaine hydrochloride (JP18) <JP> |
| Proxymetacaine |
| Proxymetacaine (INN) |
| Proparacaine hydrochloride (USP) <US> |
| p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN); Diethylaminoethyl p-butylaminobenzoate hydrochloride (JAN) |