AR225031A1 - COMPOUND OF PENICILANIC ACID 1,1-DIOXIDE, WITHOUT THERAPEUTIC ACTIVITY, USEFUL AS INTERMEDIARIES TO DEVELOP BETA-LACTAMASE INHIBITORS AND PROCEDURE TO PRODUCE SUCH BETA-LACTAMASE INHIBITORS, BASED ON SUCH INTERIODES - Google Patents

COMPOUND OF PENICILANIC ACID 1,1-DIOXIDE, WITHOUT THERAPEUTIC ACTIVITY, USEFUL AS INTERMEDIARIES TO DEVELOP BETA-LACTAMASE INHIBITORS AND PROCEDURE TO PRODUCE SUCH BETA-LACTAMASE INHIBITORS, BASED ON SUCH INTERIODES

Info

Publication number
AR225031A1
AR225031A1 AR280148A AR28014880A AR225031A1 AR 225031 A1 AR225031 A1 AR 225031A1 AR 280148 A AR280148 A AR 280148A AR 28014880 A AR28014880 A AR 28014880A AR 225031 A1 AR225031 A1 AR 225031A1
Authority
AR
Argentina
Prior art keywords
beta
lactamase inhibitors
interiodes
intermediaries
dioxide
Prior art date
Application number
AR280148A
Other languages
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR225031A1 publication Critical patent/AR225031A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AR280148A 1979-03-05 1980-03-03 COMPOUND OF PENICILANIC ACID 1,1-DIOXIDE, WITHOUT THERAPEUTIC ACTIVITY, USEFUL AS INTERMEDIARIES TO DEVELOP BETA-LACTAMASE INHIBITORS AND PROCEDURE TO PRODUCE SUCH BETA-LACTAMASE INHIBITORS, BASED ON SUCH INTERIODES AR225031A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1780879A 1979-03-05 1979-03-05
US1781079A 1979-03-05 1979-03-05

Publications (1)

Publication Number Publication Date
AR225031A1 true AR225031A1 (en) 1982-02-15

Family

ID=26690337

Family Applications (1)

Application Number Title Priority Date Filing Date
AR280148A AR225031A1 (en) 1979-03-05 1980-03-03 COMPOUND OF PENICILANIC ACID 1,1-DIOXIDE, WITHOUT THERAPEUTIC ACTIVITY, USEFUL AS INTERMEDIARIES TO DEVELOP BETA-LACTAMASE INHIBITORS AND PROCEDURE TO PRODUCE SUCH BETA-LACTAMASE INHIBITORS, BASED ON SUCH INTERIODES

Country Status (36)

Country Link
KR (1) KR850001339B1 (en)
AR (1) AR225031A1 (en)
AT (1) AT366693B (en)
AU (1) AU522572B2 (en)
BG (1) BG33292A3 (en)
CH (1) CH644608A5 (en)
CS (1) CS215130B2 (en)
DD (1) DD149367A5 (en)
DE (1) DE3008257C2 (en)
DK (2) DK159852C (en)
EG (1) EG14437A (en)
ES (1) ES8103094A1 (en)
FI (1) FI70024C (en)
FR (1) FR2450836B1 (en)
GB (1) GB2045755B (en)
GR (1) GR67234B (en)
HK (1) HK66587A (en)
HU (1) HU186304B (en)
IE (1) IE49535B1 (en)
IL (1) IL59515A (en)
IN (1) IN153685B (en)
IT (1) IT1130300B (en)
KE (1) KE3464A (en)
LU (1) LU82215A1 (en)
MX (1) MX6032E (en)
MY (1) MY8500319A (en)
NL (1) NL180317C (en)
NO (2) NO800618L (en)
PL (1) PL125197B1 (en)
PT (1) PT70897A (en)
RO (1) RO80112A (en)
SE (2) SE449103B (en)
SG (1) SG55884G (en)
SU (1) SU1192626A3 (en)
UA (1) UA6342A1 (en)
YU (1) YU42328B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419284A (en) * 1981-03-23 1983-12-06 Pfizer Inc. Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide
IN159362B (en) * 1981-03-23 1987-05-09 Pfizer
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
IT1190897B (en) * 1982-06-29 1988-02-24 Opos Biochimica Srl PROCEDURE FOR THE PREPARATION OF THE 1-ETHOXYCARBONYLOXYETHYL ACID ACID 6- (D (-) - ALPHA AMINOALPHA-PHENYLACETAMIDE) -PENICILLANIC
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
EP0139047A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the preparation of 6,6-dibromopenicillanic acid 1,1-dioxide
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4596677A (en) * 1984-04-06 1986-06-24 Bristol-Myers Company Anhydropenicillin intermediates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (en) * 1977-06-07 1982-04-03 Pfizer
CA1158639A (en) * 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
EP0013617B1 (en) * 1979-01-10 1984-07-04 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives

Also Published As

Publication number Publication date
ATA119080A (en) 1981-09-15
GB2045755B (en) 1983-01-26
GB2045755A (en) 1980-11-05
SE8603309L (en) 1986-08-04
BG33292A3 (en) 1983-01-14
NO800618L (en) 1980-09-08
IE800429L (en) 1980-09-05
NO823127L (en) 1980-09-08
DE3008257A1 (en) 1980-09-11
SE8000512L (en) 1980-09-06
ES489185A0 (en) 1981-02-16
HK66587A (en) 1987-09-25
DD149367A5 (en) 1981-07-08
AT366693B (en) 1982-04-26
NL180317C (en) 1987-02-02
KE3464A (en) 1984-10-12
IL59515A (en) 1983-02-23
DK145690D0 (en) 1990-06-14
PT70897A (en) 1980-04-01
DK159852B (en) 1990-12-17
EG14437A (en) 1984-09-30
GR67234B (en) 1981-06-25
YU58580A (en) 1983-02-28
HU186304B (en) 1985-07-29
IT1130300B (en) 1986-06-11
SE8603309D0 (en) 1986-08-04
FI800661A (en) 1980-09-06
NL8001285A (en) 1980-09-09
KR850001339B1 (en) 1985-09-19
FR2450836A1 (en) 1980-10-03
FI70024B (en) 1986-01-31
SU1192626A3 (en) 1985-11-15
YU42328B (en) 1988-08-31
MX6032E (en) 1984-10-04
MY8500319A (en) 1985-12-31
PL125197B1 (en) 1983-04-30
UA6342A1 (en) 1994-12-29
RO80112A (en) 1982-10-26
PL222448A1 (en) 1981-01-02
SG55884G (en) 1985-03-08
DE3008257C2 (en) 1984-03-01
DK92680A (en) 1980-09-06
FR2450836B1 (en) 1986-03-21
SE449103B (en) 1987-04-06
DK166353C (en) 1993-09-06
NL180317B (en) 1986-09-01
CH644608A5 (en) 1984-08-15
LU82215A1 (en) 1980-09-24
FI70024C (en) 1986-09-12
IE49535B1 (en) 1985-10-16
IT8020367A0 (en) 1980-03-05
AU5610480A (en) 1980-09-11
DK166353B (en) 1993-04-13
IN153685B (en) 1984-08-04
DK159852C (en) 1991-05-06
CS215130B2 (en) 1982-07-30
IL59515A0 (en) 1980-06-30
AU522572B2 (en) 1982-06-17
DK145690A (en) 1990-06-14
ES8103094A1 (en) 1981-02-16

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