DK145377C - METHOD OF ANALOGUE FOR THE PREPARATION OF N- (2'-PYRROLIDINYLMETHYL) BENZAMIDES OR ACID ADDITION SALTS OR QUATERNARY AMMONIUM SALT OR OPTICALLY ACTIVE ISOMERS THEREOF - Google Patents

METHOD OF ANALOGUE FOR THE PREPARATION OF N- (2'-PYRROLIDINYLMETHYL) BENZAMIDES OR ACID ADDITION SALTS OR QUATERNARY AMMONIUM SALT OR OPTICALLY ACTIVE ISOMERS THEREOF

Info

Publication number: DK145377C
Authority: DK; Denmark
Prior art keywords: pyrrolidinylmethyl; benzamides; analogue; preparation; quaternary ammonium
Prior art date: 1974-03-05

Application number

DK86975A

Other languages

Danish (da)

Other versions

DK86975A (en

DK145377B (en

Inventor

Gerard Bulteau

Jacques Acher

Jean-Claude Monier

Original Assignee

Soc Et Scient Et Ind

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-03-05

Filing date

1975-03-04

Publication date

1983-04-11

1974-03-05 Priority claimed from FR7407535A external-priority patent/FR2262966A1/en

1975-02-07 Priority claimed from FR7503800A external-priority patent/FR2299863B1/en

1975-03-04 Application filed by Soc Et Scient Et Ind filed Critical Soc Et Scient Et Ind

1975-11-03 Publication of DK86975A publication Critical patent/DK86975A/en

1982-11-08 Publication of DK145377B publication Critical patent/DK145377B/en

1983-04-11 Application granted granted Critical

1983-04-11 Publication of DK145377C publication Critical patent/DK145377C/en

Links

239000002253 acid Substances 0.000 title 1
229940054066 benzamide antipsychotics Drugs 0.000 title 1
150000003936 benzamides Chemical class 0.000 title 1
150000003242 quaternary ammonium salts Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
- C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D207/28—2-Pyrrolidone-5- carboxylic acids; Functional derivatives thereof, e.g. esters, nitriles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Pyrrole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK86975A 1974-03-05 1975-03-04 METHOD OF ANALOGUE FOR THE PREPARATION OF N- (2'-PYRROLIDINYLMETHYL) BENZAMIDES OR ACID ADDITION SALTS OR QUATERNARY AMMONIUM SALT OR OPTICALLY ACTIVE ISOMERS THEREOF DK145377C (en)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
FR7407535		1974-03-05
FR7407535A FR2262966A1 (en)	1974-03-05	1974-03-05	New heterocyclic benzamide and its manufacturing process
FR7503800A FR2299863B1 (en)	1975-02-07	1975-02-07	Novel substituted N- (Z-pyrrolidiny alkyl) benzamides, their derivatives and process for their preparation
FR7503800		1975-02-07

Publications (3)

Publication Number	Publication Date
DK86975A DK86975A (en)	1975-11-03
DK145377B DK145377B (en)	1982-11-08
DK145377C true DK145377C (en)	1983-04-11

Family

ID=26218210

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK86975A DK145377C (en)	1974-03-05	1975-03-04	METHOD OF ANALOGUE FOR THE PREPARATION OF N- (2'-PYRROLIDINYLMETHYL) BENZAMIDES OR ACID ADDITION SALTS OR QUATERNARY AMMONIUM SALT OR OPTICALLY ACTIVE ISOMERS THEREOF

Country Status (27)

Country	Link
JP (1)	JPS6015616B2 (en)
AR (1)	AR206621A1 (en)
AT (1)	AT358570B (en)
BG (1)	BG24666A3 (en)
CA (1)	CA1047504A (en)
CH (1)	CH605794A5 (en)
CS (1)	CS189692B2 (en)
DD (1)	DD119420A5 (en)
DE (1)	DE2507989A1 (en)
DK (1)	DK145377C (en)
EG (1)	EG12577A (en)
ES (1)	ES435274A1 (en)
FI (1)	FI750620A (en)
GB (1)	GB1466822A (en)
HK (1)	HK14078A (en)
HU (1)	HU170637B (en)
IE (1)	IE40818B1 (en)
IL (1)	IL46696A (en)
LU (1)	LU71949A1 (en)
NL (1)	NL7502608A (en)
NO (1)	NO750713L (en)
OA (1)	OA04966A (en)
PH (1)	PH14197A (en)
PL (1)	PL97091B1 (en)
RO (2)	RO72844A (en)
SE (1)	SE411754B (en)
SU (1)	SU609464A1 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NZ186175A (en) *	1977-01-27	1980-03-05	Shionogi & Co	Meta-sulphonamidobenzamide derivatives
SE8503054D0 (en) *	1985-06-19	1985-06-19	Astra Laekemedel Ab	CATECHOLCARBOXAMIDES
US4772459A (en) *	1986-09-09	1988-09-20	Erbamont, Inc.	Method for controlling emesis caused by chemotherapeutic agents and antiemetic agents useful therein
EP0314483A1 (en) *	1987-10-29	1989-05-03	Erbamont, Inc.	Preparation of benzamides
FR2699533A1 (en) *	1992-12-21	1994-06-24	Mouhtaram Mohamed	N-2-piperazinyl 4-amino:benzamide derivs. having antiemetic and antipsychotic activity

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3078497A (en) *	1960-12-29	1963-02-26	Leeds And Mieallef	Dispensing containers

1975
- 1975-02-24 IL IL46696A patent/IL46696A/en unknown
- 1975-02-25 DE DE19752507989 patent/DE2507989A1/en not_active Withdrawn
- 1975-02-26 GB GB809575A patent/GB1466822A/en not_active Expired
- 1975-03-03 EG EG109/75A patent/EG12577A/en active
- 1975-03-03 LU LU71949A patent/LU71949A1/en unknown
- 1975-03-03 AT AT160775A patent/AT358570B/en not_active IP Right Cessation
- 1975-03-03 SE SE7502342A patent/SE411754B/en not_active IP Right Cessation
- 1975-03-04 OA OA55430A patent/OA04966A/en unknown
- 1975-03-04 FI FI750620A patent/FI750620A/fi not_active Application Discontinuation
- 1975-03-04 DK DK86975A patent/DK145377C/en active
- 1975-03-04 BG BG029148A patent/BG24666A3/en unknown
- 1975-03-04 ES ES435274A patent/ES435274A1/en not_active Expired
- 1975-03-04 HU HUSO1137A patent/HU170637B/hu not_active IP Right Cessation
- 1975-03-04 CA CA221,240A patent/CA1047504A/en not_active Expired
- 1975-03-04 SU SU2112487A patent/SU609464A1/en active
- 1975-03-04 NO NO750713A patent/NO750713L/no unknown
- 1975-03-04 CS CS751445A patent/CS189692B2/en unknown
- 1975-03-04 IE IE457/75A patent/IE40818B1/en unknown
- 1975-03-05 NL NL7502608A patent/NL7502608A/en not_active Application Discontinuation
- 1975-03-05 RO RO7581558A patent/RO72844A/en unknown
- 1975-03-05 JP JP50027573A patent/JPS6015616B2/en not_active Expired
- 1975-03-05 RO RO7588831A patent/RO70647A/en unknown
- 1975-03-05 PL PL1975178533A patent/PL97091B1/en unknown
- 1975-03-05 CH CH279975A patent/CH605794A5/en not_active IP Right Cessation
- 1975-03-05 DD DD184579A patent/DD119420A5/de unknown
- 1975-04-04 AR AR257837A patent/AR206621A1/en active
1977
- 1977-08-22 PH PH20152A patent/PH14197A/en unknown
1978
- 1978-03-16 HK HK140/78A patent/HK14078A/en unknown

Also Published As

Publication number	Publication date
SU609464A3 (en)	1978-05-30
OA04966A (en)	1980-10-31
IE40818L (en)	1975-09-05
PL97091B1 (en)	1978-02-28
SE411754B (en)	1980-02-04
CA1047504A (en)	1979-01-30
PH14197A (en)	1981-03-26
HK14078A (en)	1978-03-23
DK86975A (en)	1975-11-03
AU7874075A (en)	1976-09-09
RO70647A (en)	1980-04-15
FI750620A (en)	1975-09-06
EG12577A (en)	1979-09-30
DD119420A5 (en)	1976-04-20
SE7502342L (en)	1975-09-08
BG24666A3 (en)	1978-04-12
JPS6015616B2 (en)	1985-04-20
NO750713L (en)	1975-09-08
DE2507989A1 (en)	1975-09-11
ES435274A1 (en)	1976-12-16
IL46696A0 (en)	1975-04-25
CS189692B2 (en)	1979-04-30
GB1466822A (en)	1977-03-09
IE40818B1 (en)	1979-08-29
ATA160775A (en)	1980-02-15
JPS50123668A (en)	1975-09-29
SU609464A1 (en)	1978-05-30
AR206621A1 (en)	1976-08-06
NL7502608A (en)	1975-09-09
IL46696A (en)	1978-07-31
CH605794A5 (en)	1978-10-13
DK145377B (en)	1982-11-08
AT358570B (en)	1980-09-25
LU71949A1 (en)	1976-02-04
HU170637B (en)	1977-07-28
RO72844A (en)	1981-09-24

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