DK146887C - ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES

Info

Publication number: DK146887C
Authority: DK; Denmark
Prior art keywords: thieno; preparation; benzodiazepine derivatives; analogy procedure; analogy
Prior art date: 1974-11-26

Application number

DK524175A

Other languages

Danish (da)

Other versions

DK524175A (en

DK146887B (en

Inventor

Jiban Kumar Chakrabarti

David Edward Tupper

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-11-26

Filing date

1975-11-20

Publication date

1984-07-09

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10459213&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK146887(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1975-11-20 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1976-05-27 Publication of DK524175A publication Critical patent/DK524175A/en

1979-09-07 Priority to DK375479A priority Critical patent/DK147020C/en

1984-01-30 Publication of DK146887B publication Critical patent/DK146887B/en

1984-07-09 Application granted granted Critical

1984-07-09 Publication of DK146887C publication Critical patent/DK146887C/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK524175A 1974-11-26 1975-11-20 ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES DK146887C (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DK375479A DK147020C (en)	1974-11-26	1979-09-07	THIENO (1,5) BENZODIAZEPINE COMPOUNDS FOR USE AS INTERMEDIATES

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB5124074		1974-11-26
GB51240/74A GB1533235A (en)	1974-11-26	1974-11-26	Benzodiazepine derivatives

Publications (3)

Publication Number	Publication Date
DK524175A DK524175A (en)	1976-05-27
DK146887B DK146887B (en)	1984-01-30
DK146887C true DK146887C (en)	1984-07-09

Family

ID=10459213

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK524175A DK146887C (en)	1974-11-26	1975-11-20	ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES

Country Status (30)

Country	Link
JP (1)	JPS6044314B2 (en)
AR (1)	AR221203A1 (en)
AT (1)	AT351547B (en)
AU (1)	AU506340B2 (en)
BE (1)	BE835932A (en)
BG (1)	BG29573A3 (en)
CA (1)	CA1075687A (en)
CH (2)	CH613454A5 (en)
CS (1)	CS236753B2 (en)
DD (1)	DD123343A5 (en)
DE (1)	DE2552403C2 (en)
DK (1)	DK146887C (en)
ES (1)	ES443011A1 (en)
FR (1)	FR2292479A1 (en)
GB (1)	GB1533235A (en)
HK (1)	HK58681A (en)
HU (1)	HU172493B (en)
IE (1)	IE42564B1 (en)
IL (1)	IL48502A (en)
KE (1)	KE3163A (en)
MY (1)	MY8200149A (en)
NL (1)	NL186088C (en)
NZ (1)	NZ179335A (en)
PH (2)	PH11669A (en)
PL (1)	PL100135B1 (en)
RO (1)	RO69912A (en)
SE (2)	SE421209B (en)
SU (2)	SU629879A3 (en)
YU (1)	YU298375A (en)
ZA (1)	ZA757344B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL62792A (en) *	1980-05-07	1985-02-28	Byk Gulden Lomberg Chem Fab	Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
GB9009229D0 (en) *	1990-04-25	1990-06-20	Lilly Industries Ltd	Pharmaceutical compounds
NZ247703A (en) *	1992-05-29	1995-07-26	Lilly Industries Ltd	Thienobenzdiazepine derivatives and medicaments thereof
CA2234641A1 (en) *	1995-11-01	1997-05-09	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
US6043358A (en)	1995-11-01	2000-03-28	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
EP1016664B1 (en)	1997-09-02	2003-07-02	Mitsubishi Pharma Corporation	Fused thiophene compounds and medicinal use thereof
PL199016B1 (en) *	2002-06-20	2008-08-29	Adamed Sp Z Oo	Method of manufacture of alanzapine, new derivative of n-demethyl olanzapine and method of manufacture of new derivative of n-demethyl olanzapine
SI21270A (en)	2002-07-15	2004-02-29	Krka, Tovarna Zdravil, D.D., Novo Mesto	Crystal forms of olanzapine and procedures for their preparation
DE10301923B3 (en) *	2003-01-17	2004-09-16	Krka Tovarna Zdravil, D.D.	Process and intermediates for the production of olanzapine
AR047461A1 (en) *	2004-01-27	2006-01-18	Synthon Bv	TRAINING, PURIFICATION AND USE OF N-FORMILOLANZAPINE
AR048272A1 (en)	2004-03-18	2006-04-12	Lek Pharmaceuticals	SYNTHESIS OF 2 METHYL - 4- (4- METHYL -1- PIPERAZINIL) - 10 H- TIENO (2,3-B) (1,5) BENZODIAZEPIN AND ITS SALTS, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING IT AND ITS USE IN THE MANUFACTURE OF MEDICINES FOR THE TREATMENT OF MENTAL DISEASES.
CN1980710B (en) *	2004-06-30	2013-06-12	阿特西斯公司	Substituted azepine derivatives as serotonin receptor modulators
EP2292624A1 (en)	2009-07-20	2011-03-09	LEK Pharmaceuticals d.d.	Process for the purification of olanzapine

1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/en active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
1975
- 1975-11-20 DK DK524175A patent/DK146887C/en active
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-20 IL IL48502A patent/IL48502A/en unknown
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-22 DE DE2552403A patent/DE2552403C2/en not_active Expired
- 1975-11-24 SE SE7513185A patent/SE421209B/en not_active IP Right Cessation
- 1975-11-24 CH CH1517275A patent/CH613454A5/en not_active IP Right Cessation
- 1975-11-24 NZ NZ179335A patent/NZ179335A/en unknown
- 1975-11-24 ZA ZA757344A patent/ZA757344B/en unknown
- 1975-11-24 CH CH604478A patent/CH613455A5/en not_active IP Right Cessation
- 1975-11-25 FR FR7535900A patent/FR2292479A1/en active Granted
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-25 AR AR261340A patent/AR221203A1/en active
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/en not_active Expired
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-25 RO RO7584018A patent/RO69912A/en unknown
- 1975-11-25 YU YU02983/75A patent/YU298375A/en unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/en not_active IP Right Cessation
- 1975-11-26 CS CS757991A patent/CS236753B2/en unknown
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/en not_active IP Right Cessation
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/en unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/en not_active Expired
- 1975-11-26 AT AT898275A patent/AT351547B/en not_active IP Right Cessation
- 1975-11-26 BG BG031601A patent/BG29573A3/en unknown
- 1975-11-26 PL PL1975184991A patent/PL100135B1/en unknown
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/en active
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/en not_active IP Right Cessation
1981
- 1981-09-24 KE KE3163A patent/KE3163A/en unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/en unknown
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/en unknown

Also Published As

Publication number	Publication date
DD123343A5 (en)	1976-12-12
MY8200149A (en)	1982-12-31
CS236753B2 (en)	1985-05-15
FR2292479A1 (en)	1976-06-25
CA1075687A (en)	1980-04-15
CH613454A5 (en)	1979-09-28
YU298375A (en)	1982-10-31
DE2552403C2 (en)	1986-06-19
GB1533235A (en)	1978-11-22
FR2292479B1 (en)	1978-07-28
BG29573A3 (en)	1980-12-12
AT351547B (en)	1979-07-25
SU629879A3 (en)	1978-10-25
SE429045B (en)	1983-08-08
HU172493B (en)	1978-09-28
JPS6044314B2 (en)	1985-10-02
RO69912A (en)	1980-08-15
NZ179335A (en)	1978-11-13
PH24534A (en)	1990-08-03
DK524175A (en)	1976-05-27
SE7812194L (en)	1978-11-27
ES443011A1 (en)	1977-07-01
DK146887B (en)	1984-01-30
SU626702A3 (en)	1978-09-30
IL48502A (en)	1980-01-31
ZA757344B (en)	1976-11-24
PL100135B1 (en)	1978-09-30
AU506340B2 (en)	1979-12-20
ATA898275A (en)	1979-01-15
CH613455A5 (en)	1979-09-28
KE3163A (en)	1981-10-16
IE42564L (en)	1976-05-26
BE835932A (en)	1976-05-25
NL186088C (en)	1990-09-17
AR221203A1 (en)	1981-01-15
DE2552403A1 (en)	1976-08-12
IE42564B1 (en)	1980-09-10
SE7513185L (en)	1976-05-27
SE421209B (en)	1981-12-07
PH11669A (en)	1978-05-19
JPS5176296A (en)	1976-07-01
IL48502A0 (en)	1976-01-30
NL186088B (en)	1990-04-17
AU8685875A (en)	1977-05-26
HK58681A (en)	1981-12-04
NL7513833A (en)	1976-05-31

Publication	Publication Date	Title
DK487476A (en)	1977-04-30	PROCEDURE FOR THE PREPARATION OF IMIDAZOLIDINES
DK157487C (en)	1990-06-11	ANALOGY PROCEDURE FOR THE PREPARATION OF PROLINE DERIVATIVES.
DK149107C (en)	1986-06-09	ANALOGY PROCEDURE FOR THE PREPARATION OF QUINAZOLON DERIVATIVES
DK146205C (en)	1983-12-27	ANALOGY PROCEDURE FOR THE PREPARATION OF 8ALFA ERGOLIN-I DERIVATIVES
DK55477A (en)	1977-08-11	PROCEDURE FOR THE PREPARATION OF 1,2-DITHIOL DERIVATIVES
DK146887C (en)	1984-07-09	ANALOGY PROCEDURE FOR THE PREPARATION OF THIENO (1,5) BENZODIAZEPINE DERIVATIVES
DK55677A (en)	1977-08-11	PROCEDURE FOR THE PREPARATION OF 1,2-DITHIOL DERIVATIVES
DK164376A (en)	1976-10-26	PROCEDURE FOR THE PREPARATION OF 3,4-DIHYDROSPIRO-2H-1,3-BENZOXAZINES
DK554076A (en)	1977-06-12	PROCEDURE FOR THE PREPARATION OF 3,4I-DIDEOXYCANAMYCINE]
DK143902C (en)	1982-04-13	ANALOGY PROCEDURE FOR THE PREPARATION OF 8ALFA ERGOLIN-I DERIVATIVES
DK148139C (en)	1985-09-30	ANALOGY PROCEDURE FOR THE PREPARATION OF 5-BENZYL-2-OXAZOLIDE UNDERTIVES
DK154970C (en)	1989-06-12	ANALOGY PROCEDURE FOR THE PREPARATION OF CARBOSTYRIC DERIVATIVES
DK356375A (en)	1976-02-07	PROCEDURE FOR THE PREPARATION OF 2-THIOL-4,5-DIPHENYLOXAZOLE-S DERIVATIVES
SE419983B (en)	1981-09-07	PROCEDURE FOR THE PREPARATION OF FINE-CORN, SOLID CYANURCHLORIDE
DK143757C (en)	1982-03-22	ANALOGY PROCEDURE FOR THE PREPARATION OF 16,16-DISUBSTITUTED 3-OXOANDROSTEN
DK148098C (en)	1985-07-29	ANALOGY PROCEDURE FOR THE PREPARATION OF DAUNOMYCIN DERIVATIVES
DK153479C (en)	1988-11-28	ANALOGY PROCEDURE FOR THE PREPARATION OF 1,4-BENZODIAZEPIN-2-ON DERIVATIVES
DK146629C (en)	1984-04-30	ANALOGY PROCEDURE FOR THE PREPARATION OF DEPOTTEROID EASTERS
DK155316C (en)	1989-08-14	ANALOGY PROCEDURE FOR THE PREPARATION OF OMEGA-NOR-CYCLOALKYL-13,14-DEHYDROPROSTAGLANDINES
DK147070C (en)	1984-09-10	ANALOGY PROCEDURE FOR THE PREPARATION OF 13,14-DEHYDRO-11-DEOXY PROSTAGLANDINES
DK227476A (en)	1976-11-29	PROCEDURE FOR THE PREPARATION OF 4,5,6,7-TETRAHYDRO-THIENO (3,2-C) -PYRIDINE DERIVATIVES
DK416476A (en)	1977-03-25	PROCEDURE FOR THE PREPARATION OF DIAZEPINE DERIVATIVES
DK142845C (en)	1981-08-31	ANALOGY PROCEDURE FOR THE PREPARATION OF IMIDAZOLD DERIVATIVES
DK149803C (en)	1987-04-06	PROCEDURE FOR THE PREPARATION OF 1,2-DICHLORETHAN
DK544476A (en)	1977-06-06	PROCEDURE FOR THE PREPARATION OF DIFLUOROMETHYL-1,2,2-TRIFLUOROETHYLETHER