DK297486A - benzoxazinone derivatives - Google Patents

benzoxazinone derivatives Download PDF

Info

Publication number: DK297486A
Authority: DK; Denmark
Prior art keywords: benzoxazinone derivatives; benzoxazinone; derivatives
Prior art date: 1985-06-25

Application number

DK297486A

Other languages

Danish (da)

Other versions

DK297486D0 (en

Inventor

Alexander Krantz

Robin W Spencer

Tim Tam

Teng J Liak

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-25

Filing date

1986-06-24

Publication date

1986-12-26

1986-06-24 Application filed by Syntex Inc filed Critical Syntex Inc

1986-06-24 Publication of DK297486D0 publication Critical patent/DK297486D0/en

1986-12-26 Publication of DK297486A publication Critical patent/DK297486A/en

Links

HQQTZCPKNZVLFF-UHFFFAOYSA-N 4h-1,2-benzoxazin-3-one Chemical class C1=CC=C2ONC(=O)CC2=C1 HQQTZCPKNZVLFF-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
- C07F9/6533—Six-membered rings
- C07F9/65335—Six-membered rings condensed with carbocyclic rings or carbocyclic ring systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DK297486A 1985-06-25 1986-06-24 benzoxazinone derivatives DK297486A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/748,631 US4665070A (en)	1985-06-25	1985-06-25	2-oxy-4H-3,1-benzoxazin-4-ones and pharmaceutical use

Publications (2)

Publication Number	Publication Date
DK297486D0 DK297486D0 (en)	1986-06-24
DK297486A true DK297486A (en)	1986-12-26

Family

ID=25010264

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK297486A DK297486A (en)	1985-06-25	1986-06-24	benzoxazinone derivatives

Country Status (13)

Country	Link
US (1)	US4665070A (en)
EP (1)	EP0206323A1 (en)
JP (1)	JPS6230770A (en)
KR (1)	KR900004319B1 (en)
AU (2)	AU599320B2 (en)
CA (1)	CA1270487A (en)
DK (1)	DK297486A (en)
ES (4)	ES8802223A1 (en)
FI (1)	FI862691A (en)
HU (1)	HU196772B (en)
IL (1)	IL79222A0 (en)
NO (1)	NO163486C (en)
ZA (1)	ZA864715B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4745116A (en) *	1985-06-25	1988-05-17	Syntex (U.S.A.) Inc.	2-oxy-4H-3,1-benzoxazin-4-ones and related compounds and pharmaceutical use
CA1309556C (en) *	1987-06-09	1992-10-27	Masayuki Kokubo	4h-3,1-benzoxazin-4-one compounds and pharmaceutical composition thereoffor the inhibition of serine proteases
EP0480044A4 (en) *	1990-03-30	1993-06-09	Japan Tobacco Inc.	Novel 4h-3,1-benzoxazin-4-one derivative
US5985872A (en) *	1995-05-24	1999-11-16	G.D. Searle & Co.	2-amino-benzoxazinones for the treatment of viral infections
FR2763944B1 (en) *	1997-06-03	2000-12-15	Centre Nat Rech Scient	NOVEL COUMARIN DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS DRUGS AS PROTEASE INHIBITORS
US6180625B1 (en)	1998-03-24	2001-01-30	Novo Nordisk A/S	Heterocyclic compounds regulating clotting
WO1999048878A1 (en) *	1998-03-24	1999-09-30	Novo Nordisk A/S	Heterocyclic compounds regulating clotting
WO2000030646A1 (en) *	1998-11-26	2000-06-02	Novo Nordisk A/S	Heterocyclic compounds regulating clotting
GB9900416D0 (en)	1999-01-08	1999-02-24	Alizyme Therapeutics Ltd	Inhibitors
AR022204A1 (en) *	1999-01-08	2002-09-04	Norgine Bv	COMPOUND, PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION AND EDIBLE PRODUCT THAT UNDERSTANDS IT.
WO2001018181A2 (en) *	1999-09-10	2001-03-15	The Procter & Gamble Company	Enzyme inhibitors
CA2524882A1 (en) *	2003-05-06	2004-11-25	Cytovia, Inc.	Protease inhibitors for coronaviruses and sars-cov and the use thereof
JP5273587B2 (en) *	2006-11-22	2013-08-28	味の素株式会社	Process for producing phenylalanine derivative having quinazolinedione skeleton and production intermediate
JP2010254623A (en) *	2009-04-24	2010-11-11	Takeda Chem Ind Ltd	Crystal of benzoxazinone compound

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU173974B (en) *	1971-08-30	1979-10-28	Chinoin Gyogyszer Es Vegyeszet	Process for preparing 3,1-benzoxazin-4-one derivatives

1985
- 1985-06-25 US US06/748,631 patent/US4665070A/en not_active Expired - Fee Related
1986
- 1986-06-24 KR KR1019860005053A patent/KR900004319B1/en not_active IP Right Cessation
- 1986-06-24 IL IL79222A patent/IL79222A0/en unknown
- 1986-06-24 ZA ZA864715A patent/ZA864715B/en unknown
- 1986-06-24 NO NO862534A patent/NO163486C/en unknown
- 1986-06-24 AU AU59150/86A patent/AU599320B2/en not_active Ceased
- 1986-06-24 DK DK297486A patent/DK297486A/en not_active Application Discontinuation
- 1986-06-24 CA CA000512310A patent/CA1270487A/en not_active Expired - Fee Related
- 1986-06-24 JP JP61149323A patent/JPS6230770A/en active Pending
- 1986-06-24 HU HU862647A patent/HU196772B/en not_active IP Right Cessation
- 1986-06-24 EP EP86108617A patent/EP0206323A1/en not_active Ceased
- 1986-06-24 ES ES556514A patent/ES8802223A1/en not_active Expired
- 1986-06-24 FI FI862691A patent/FI862691A/en not_active Application Discontinuation
1987
- 1987-09-16 ES ES557730A patent/ES8801806A1/en not_active Expired
- 1987-09-16 ES ES557732A patent/ES8801808A1/en not_active Expired
- 1987-09-16 ES ES557731A patent/ES8801807A1/en not_active Expired
1990
- 1990-02-07 AU AU49120/90A patent/AU4912090A/en not_active Abandoned

Also Published As

Publication number	Publication date
AU4912090A (en)	1990-05-31
ES557730A0 (en)	1988-03-01
FI862691A (en)	1986-12-26
HUT41750A (en)	1987-05-28
AU5915086A (en)	1987-01-08
ES8802223A1 (en)	1988-05-01
ES8801808A1 (en)	1988-03-01
KR900004319B1 (en)	1990-06-22
AU599320B2 (en)	1990-07-19
JPS6230770A (en)	1987-02-09
EP0206323A1 (en)	1986-12-30
ES8801806A1 (en)	1988-03-01
CA1270487A (en)	1990-06-19
ES557732A0 (en)	1988-03-01
HU196772B (en)	1989-01-30
NO862534D0 (en)	1986-06-24
ZA864715B (en)	1988-02-24
US4665070A (en)	1987-05-12
IL79222A0 (en)	1986-09-30
ES556514A0 (en)	1988-05-01
NO163486B (en)	1990-02-26
NO862534L (en)	1986-12-29
ES557731A0 (en)	1988-03-01
FI862691A0 (en)	1986-06-24
DK297486D0 (en)	1986-06-24
KR870000310A (en)	1987-02-17
NO163486C (en)	1990-06-13
ES8801807A1 (en)	1988-03-01

Legal Events

Date	Code	Title	Description
1992-02-24	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
DK263587A (en)	1987-11-24	IMIDAZOQUINOLINYLETHERY DERIVATIVES
DK82087A (en)	1987-09-12	PYROCATECHAL DERIVATIVES
ATE49403T1 (en)	1990-01-15	N-ARALKYLPIPERIDINEMETHANOL DERIVATIVES.
DK69887A (en)	1987-08-13	DICHLORANILINE DERIVATIVES
ATA312487A (en)	1993-05-15	TETRAHYDROCARBAZOLONE DERIVATIVES
DE3675232D1 (en)	1990-12-06	PYRIDE DERIVATIVES.
DE3678805D1 (en)	1991-05-23	INDOLDER DERIVATIVES.
DK693587A (en)	1988-07-01	ALKANSULPHONANILIDE DERIVATIVES
DK297486D0 (en)	1986-06-24	benzoxazinone derivatives
DE3680067D1 (en)	1991-08-08	FLUORPHENYLCYCLOHEXANE DERIVATIVES.
DK109186A (en)	1986-09-13	DIHYDROPYRIDAZINON DERIVATIVES
ATE41655T1 (en)	1989-04-15	PHENAETHANOLAMINE DERIVATIVES.
DK691287D0 (en)	1987-12-29	5-FLOURURACIL DERIVATIVES
DK491786D0 (en)	1986-10-14	DICHLORANILINE DERIVATIVES
BR8606663A (en)	1987-08-11	TRIAZOLYL-QUINOLINE DERIVATIVES
DK444687A (en)	1988-02-28	ALFA-SUBSTITUTED KETONITRON DERIVATIVES
DK556386D0 (en)	1986-11-20	QUINILIN DERIVATIVES
DK303886A (en)	1986-12-29	SECOCANTHIN DERIVATIVES
DK229887A (en)	1987-11-09	ALKENAMIDE DERIVATIVES
DK619187A (en)	1988-05-28	ISOINDOLD DERIVATIVES
DK440687D0 (en)	1987-08-24	BICYCLOOCTAN DERIVATIVES
DE3662889D1 (en)	1989-05-24	TETRAHYDROFURANCARBOXYLIC-ACID DERIVATIVES
KR880700821A (en)	1988-04-12	De-deoxyteicoplanin derivatives
DK435087A (en)	1988-03-11	ISOPRENDER DERIVATIVES
DK440787D0 (en)	1987-08-24	BICYCLOOCTAN DERIVATIVES