GB1536282A - Thiazolylacetic acid derivatives - Google Patents

Thiazolylacetic acid derivatives

Info

Publication number: GB1536282A
Authority: GB; United Kingdom
Prior art keywords: acid derivatives; thiazolylacetic acid; thiazolylacetic; derivatives; acid
Prior art date: 1974-12-19
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

GB51582/75A

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Takeda Pharmaceutical Co Ltd

Original Assignee

Takeda Chemical Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-12-19

Filing date

1975-12-17

Publication date

1978-12-20

1975-12-17 Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd

1978-12-20 Publication of GB1536282A publication Critical patent/GB1536282A/en

Status Expired legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/34—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Thiazole And Isothizaole Compounds (AREA)
Cephalosporin Compounds (AREA)

GB51582/75A 1974-12-19 1975-12-17 Thiazolylacetic acid derivatives Expired GB1536282A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP49146567A JPS5760345B2 (en)	1974-12-19	1974-12-19

Publications (1)

Publication Number	Publication Date
GB1536282A true GB1536282A (en)	1978-12-20

Family

ID=15410584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
GB51582/75A Expired GB1536282A (en)	1974-12-19	1975-12-17	Thiazolylacetic acid derivatives

Country Status (6)

Country	Link
US (1)	US4355160A (en)
JP (1)	JPS5760345B2 (en)
GB (1)	GB1536282A (en)
HK (1)	HK2382A (en)
MY (1)	MY8200220A (en)
ZA (1)	ZA757892B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2714880A1 (en) *	1977-04-02	1978-10-26	Hoechst Ag	CEPHEMDER DERIVATIVES AND PROCESS FOR THEIR PRODUCTION
US5089490A (en) *	1977-04-02	1992-02-18	Hoechst Aktiengesellschaft	Cephem derivatives
JPS57154175A (en) *	1981-03-16	1982-09-22	Mitsui Toatsu Chem Inc	2-thiazoleamine derivative, its preparation, and drug composition comprising it
JPS5979935U (en) *	1982-11-20	1984-05-30	日本開閉器工業株式会社	small tilt switch
US4788185A (en) *	1984-04-23	1988-11-29	Takeda Chemical Industries, Ltd.	Cephalosporin compounds
JPS6310795A (en) *	1986-03-25	1988-01-18	Takeda Chem Ind Ltd	Selective herbicidal compound
FR2621589B1 (en) *	1987-10-08	1990-03-02	Sanofi Sa	CEPHALOSPORIN DERIVATIVES WITH IMPROVED PHARMACOKINETICS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DE3804841A1 (en) *	1988-02-17	1989-08-31	Hoechst Ag	CEPHALOSPORINE DERIVATIVES AND METHOD FOR THEIR PRODUCTION
DE3919259A1 (en) *	1989-06-13	1990-12-20	Hoechst Ag	CRYSTALLINE CEPHEM ACID ADDITION SALTS AND METHOD FOR THE PRODUCTION THEREOF
YU48484B (en) *	1991-05-24	1998-09-18	Hoechst Aktiengesellschaft	Crystal acid addition salts diastereometric pure 1-(-2,2-dimethylpropyonyloxy)-ethylesters 3-pephem-4-carbonic acid
DE59209994D1 (en) *	1991-09-07	2004-04-29	Aventis Pharma Gmbh	Diastereomer of 3-cephem-4-carboxylic acid 1 - (- isopropoxycarbonyloxy) ethyl ester and process for its preparation
TW212181B (en) *	1992-02-14	1993-09-01	Hoechst Ag
EP0570849B1 (en) *	1992-05-21	1998-03-25	Hoechst Aktiengesellschaft	Process for the cleavage of cephalosporin prodrug esters to 7-amino-3-methoxymethylceph-3-em-4-carboxylic acid
CN114031575B (en) *	2021-12-15	2023-09-12	山东金城医药化工有限公司	Preparation method of ethyl northioxomate

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1364453A (en) *	1970-11-06	1974-08-21	Gist Brocades Nv	Penicillanic and cepholosporanic acid derivatives
US3855213A (en) *	1971-02-18	1974-12-17	Smith Kline French Lab	3-heterocyclic thiomethyl-cephalosporins
US4024134A (en) *	1971-01-29	1977-05-17	Glaxo Laboratories Limited	Syn isomers of cephalosporins having α-hydroximino- or α-acyloxyiminoacylamido groups at position-7
US3971778A (en) *	1972-05-12	1976-07-27	Glaxo Laboratories Limited	Cephalosporins having (α-etherified oximino)acylamido groups at the 7-position
US4024133A (en) *	1971-05-14	1977-05-17	Glaxo Laboratories Limited	7β-[2-Etherified oximino-2-(thienyl-,furyl- or pyridylacetamido)]cephalosporins
US4024137A (en) *	1971-05-14	1977-05-17	Glaxo Laboratories Limited	7β-[2-Etherified oximino-2-(phenyl- or naphthylacetamido)] cephalosporins
US3966717A (en) *	1971-05-14	1976-06-29	Glaxo Laboratories Limited	7-β-Acylamido-3-carbamoyloxymethylceph-3-em-4-carboxylic acids and salts thereof
US3974153A (en) *	1971-05-14	1976-08-10	Glaxo Laboratories Limited	7-Hydrocarbonoxy imino-acetamido-3-carbamoyloxy methylceph-3-em-4 carboxylic acids
YU36181B (en) *	1971-11-29	1982-02-25	Merck & Co Inc	Process for obtaining 7-(2-thienylacetamido)-7-methoxy-3-carbamoyloxymethyl-3-cephem-4-carboxylates
US4032521A (en) *	1972-12-29	1977-06-28	Merck & Co., Inc.	Cephalosporin phosphonic acid, sulfonic acid and sulfonamide compounds
DE2512284A1 (en) *	1974-03-28	1975-10-09	Fujisawa Pharmaceutical Co	CEPHALOSPORANIC ACID DERIVATIVES, PROCESS FOR THEIR MANUFACTURING AND PHARMACEUTICAL PRODUCTS CONTAINING THEM
DK154939C (en) *	1974-12-19	1989-06-12	Takeda Chemical Industries Ltd	METHOD OF ANALOGUE FOR THE PREPARATION OF THIAZOLYLACETAMIDO-CEPHEM COMPOUNDS OR PHARMACEUTICAL ACCEPTABLE SALTS OR ESTERS THEREOF
US4203899A (en) *	1974-12-19	1980-05-20	Takeda Chemical Industries, Ltd.	Thiazolylacetamido compounds
DE2760123C2 (en) *	1976-01-23	1986-04-30	Roussel-Uclaf, Paris	7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporanic acids, their preparation and pharmaceutical compositions containing them
JPS6011713B2 (en) *	1976-09-08	1985-03-27	武田薬品工業株式会社	Cephalosporin derivatives and their production method
JPS53101393A (en) *	1977-02-17	1978-09-04	Takeda Chem Ind Ltd	Cephalosporin derivatives and process for their preparation
US4200745A (en) *	1977-12-20	1980-04-29	Eli Lilly And Company	7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins

1974
- 1974-12-19 JP JP49146567A patent/JPS5760345B2/ja not_active Expired
1975
- 1975-12-17 GB GB51582/75A patent/GB1536282A/en not_active Expired
- 1975-12-19 ZA ZA757892A patent/ZA757892B/en unknown
1981
- 1981-03-04 US US06/240,466 patent/US4355160A/en not_active Expired - Lifetime
1982
- 1982-01-14 HK HK23/82A patent/HK2382A/en unknown
- 1982-12-30 MY MY220/82A patent/MY8200220A/en unknown

Also Published As

Publication number	Publication date
MY8200220A (en)	1982-12-31
JPS5175066A (en)	1976-06-29
HK2382A (en)	1982-01-22
ZA757892B (en)	1976-11-24
JPS5760345B2 (en)	1982-12-18
US4355160A (en)	1982-10-19

Legal Events

Date	Code	Title	Description
1979-04-11	PS	Patent sealed [section 19, patents act 1949]
1996-01-17	PE20	Patent expired after termination of 20 years	Effective date: 19951216

Publication	Publication Date	Title
GB1536283A (en)	1978-12-20	Alpha-protected oxyimino-beta-oxo-ypsilon-halogeno-butyric acid derivatives
ZA751391B (en)	1976-10-27	16-oxygenated prostanoic acid derivatives
GB1516656A (en)	1978-07-05	3-sulphonyloxy-cephem-4-carboxylic acid derivatives
AU521892B2 (en)	1982-05-06	Sulphamoylbenzoic acid derivatives
IL46341A0 (en)	1975-03-13	Alpha-aryl-4-substituted piperidinoalkanol derivatives
MY8200220A (en)	1982-12-31	Thiazolylazetic acid derivatives
ZA757290B (en)	1976-11-24	Furanhydroxamic acid derivatives
AU8504375A (en)	1977-03-31	Naphthenohydroxamic acid
AU8794575A (en)	1977-07-07	Phenylacetic acid derivatives
GB1539180A (en)	1979-01-31	1-cyclopentene-1-propanoic acid derivatives
ZA752022B (en)	1976-02-25	Prostanoic acid derivatives
ZA755543B (en)	1976-07-28	Thiomethylcephem derivatives
IL56863A0 (en)	1979-05-31	7-cyclopentyl-heptanoic acid derivatives
AU7903975A (en)	1976-09-16	Indolylacetyl-amino acid derivatives
ZA754128B (en)	1976-06-30	Monochromone-2-carboxylic acid
AU502146B2 (en)	1979-07-12	11-epi-prostanoic acid derivatives
NZ179201A (en)	1978-06-02	2(w-aminoalkyl)isoindol-i-ylcarboxylic acid derivatives
AU8692375A (en)	1977-06-02	Prostenoic acid derivatives
MY7800453A (en)	1978-12-31	2-chloroethananephosphonic acid derivatives
GB1519187A (en)	1978-07-26	Cephalosporanic acid derivatives
GB1535217A (en)	1978-12-13	20-alkoxy-16-alkyl-prostadienoic acid derivatives
JPS51138693A (en)	1976-11-30	Isoklabaranic acid derivative
ZA754492B (en)	1976-06-30	Prostanoic acid derivatives
ZA754721B (en)	1976-07-28	Prostanoic acid derivatives
GB1523278A (en)	1978-08-31	Penicillanic acid derivatives