MY115416A - Quinolone-and naphthyridone-carboxylic acid derivatives - Google Patents

Quinolone-and naphthyridone-carboxylic acid derivatives

Info

Publication number
MY115416A
MY115416A MYPI93000039A MYPI9300039A MY115416A MY 115416 A MY115416 A MY 115416A MY PI93000039 A MYPI93000039 A MY PI93000039A MY PI9300039 A MYPI9300039 A MY PI9300039A MY 115416 A MY115416 A MY 115416A
Authority
MY
Malaysia
Prior art keywords
carboxylic acid
acid derivatives
naphthyridone
quinolone
antibacterical
Prior art date
Application number
MYPI93000039A
Inventor
Uwe Dr Petersen
Andreas Dr Krebs
Thomas Dr Philipps
Klaus Dr Grohe
Klaus-Dieter Dr Bremm
Rainer Dr Endermann
Karl-Georg Dr Metzger
Ingo Dr Haller
Thomas Dr Schenke
Original Assignee
Bayer Schering Pharma Aktiemgesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27203290&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MY115416(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE4200414A external-priority patent/DE4200414A1/en
Priority claimed from DE4208789A external-priority patent/DE4208789A1/en
Priority claimed from DE4208792A external-priority patent/DE4208792A1/en
Application filed by Bayer Schering Pharma Aktiemgesellschaft filed Critical Bayer Schering Pharma Aktiemgesellschaft
Publication of MY115416A publication Critical patent/MY115416A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Fodder In General (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Apparatus For Disinfection Or Sterilisation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

THE INVENTION RELATES TO NEW QUINOLONE- AND NAPHTHYRIDONE CARBOXYLIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND ALSO ANTIBACTERICAL AGENTS AND FEED ADDITIVES CONTAINING THEM.
MYPI93000039A 1992-01-10 1993-01-10 Quinolone-and naphthyridone-carboxylic acid derivatives MY115416A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE4200414A DE4200414A1 (en) 1992-01-10 1992-01-10 New quinoline and naphthyridinone-carboxylic acid derivs.
DE4208789A DE4208789A1 (en) 1992-03-19 1992-03-19 New quinoline and naphthyridinone-carboxylic acid derivs.
DE4208792A DE4208792A1 (en) 1992-03-19 1992-03-19 New quinoline and naphthyridinone-carboxylic acid derivs.

Publications (1)

Publication Number Publication Date
MY115416A true MY115416A (en) 2003-06-30

Family

ID=27203290

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI93000039A MY115416A (en) 1992-01-10 1993-01-10 Quinolone-and naphthyridone-carboxylic acid derivatives

Country Status (16)

Country Link
EP (1) EP0550903A1 (en)
JP (3) JPH05271229A (en)
KR (1) KR100251886B1 (en)
CN (3) CN1043142C (en)
AU (1) AU669502B2 (en)
CA (1) CA2086914C (en)
CZ (1) CZ289076B6 (en)
FI (3) FI104174B (en)
HU (1) HU219488B (en)
MX (1) MX9207604A (en)
MY (1) MY115416A (en)
NO (1) NO301420B1 (en)
NZ (1) NZ245640A (en)
PL (1) PL174853B1 (en)
SK (3) SK285223B6 (en)
TW (1) TW209865B (en)

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US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
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IL142642A0 (en) * 1998-11-10 2002-03-10 Bayer Ag Pharmaceutical moxifloxacin preparation
CN1343128B (en) 1999-03-17 2010-04-21 第一制药株式会社 Medicinal compositions
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DE19931115A1 (en) * 1999-07-06 2001-01-11 Bayer Ag Racemization of R, S-dioxo-benzylpyrrolopiperidine
DE19962470A1 (en) * 1999-12-22 2001-07-12 Schulz Hans Herrmann Use of chemotherapy drugs
DE10226923A1 (en) * 2002-06-17 2003-12-24 Bayer Ag Process for the enantiomer enrichment of cis-8-benzyl-7,9-dioxo-2,8-diazabicyclo [4.3.0] nonane
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US7759362B2 (en) 2004-04-21 2010-07-20 Institut Of Medicinal Biotechnology Chinese Academy Of Medical Sciences Quinolonecarboxylic acid compounds, preparation methods and pharmaceutical uses thereof
CN1244582C (en) * 2004-04-21 2006-03-08 中国医学科学院医药生物技术研究所 Quinolone carboxylic acid compound and its preparation method and medical application
ES2284380B1 (en) * 2006-03-10 2008-11-01 Quimica Sintetica S.A. PROCEDURE FOR THE PREPARATION OF MOXIFLOXACINO AND MOXIFLOXACINO CHLORHYDRATE.
ATE446946T1 (en) 2006-06-27 2009-11-15 Sandoz Ag NEW PROCESS FOR PRODUCING SALT
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WO2008059521A2 (en) * 2006-11-14 2008-05-22 Msn Laboratories Limited Novel process for the preparation of moxifloxacin hydrochloride and a novel polymorph of moxifloxacin
US7692015B2 (en) 2007-01-05 2010-04-06 Zheqing Wang Economical process for preparing (S, S)-2, 8-diazabicyclo[4.3.0]nonane and its enantiomer
WO2008102188A1 (en) 2007-02-22 2008-08-28 Tibor Nagy Procedure to manufacture and use beer and other types liquids treated with neodimium magnet
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WO2010122774A1 (en) * 2009-04-20 2010-10-28 株式会社カネカ Processes for producing (1s,6s)- or (1r,6r)-cis-2,8-diazabicyclo[4.3.0]nonane and intermediate thereof
IT1398952B1 (en) * 2010-03-19 2013-03-28 F S I Fabbrica Italiana Sint PROCESS OF PREPARATION OF MOXIFLOXACINE AND ITS SALTS
CN101941969B (en) * 2010-09-30 2012-05-23 江苏正大丰海制药有限公司 Preparation method of moxifloxacin hydrochloride
CN102675307A (en) * 2011-03-17 2012-09-19 苏州中科天马肽工程中心有限公司 Method for preparing chiral compound 8-phenethyl-2,8-diazabicyclo[4.3.0]nonane
CN102675308A (en) * 2011-03-17 2012-09-19 苏州中科天马肽工程中心有限公司 Method for preparing 8-benzyl-2,8-diazabicyclo(4.3.0) nonane
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CN103044418B (en) * 2011-10-14 2015-02-04 上海朴颐化学科技有限公司 Asymmetric synthesis method, relevant raw materials and preparation method of (S,S)-2,8-diazabicyclo[4,3,0] nonane
CN102408427B (en) * 2011-10-22 2012-12-12 浙江普洛康裕制药有限公司 Preparation method for moxifloxacin intermediate (1S, 6R)-8-benzyl-7, 9-dioxy-2, 8-diazabicyclo [4.3.0] nonane
BRPI1106900A2 (en) 2011-12-26 2013-11-05 Ems Sa SOLID PHARMACEUTICAL COMPOSITION UNDERSTANDING ANTIBOTH FAMILY OF QUINOLONES AND THE PROCESS OF OBTAINING THEM
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CN103012452B (en) * 2012-12-25 2015-12-02 浙江新和成股份有限公司 The preparation method of a kind of Moxifloxacin and hydrochloride thereof
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CN108872413B (en) * 2018-04-27 2021-06-08 山东齐都药业有限公司 Method for detecting enantiomer content in (S, S) -2, 8-diazabicyclo [4,3,0] nonane
CN110627768B (en) * 2018-06-22 2021-11-09 扬子江药业集团有限公司 Preparation method of moxifloxacin degradation impurity J
CN110183445B (en) * 2019-06-28 2021-08-24 昆明学院 Synthetic method of moxifloxacin and its derivatives
RU2713932C1 (en) * 2019-10-31 2020-02-11 федеральное государственное автономное образовательное учреждение высшего образования "Казанский (Приволжский) федеральный университет" (ФГАОУ ВО КФУ) Fluoroquinolone compounds based on pyridoxine derivatives, having antibacterial properties
CN112939849B (en) * 2019-12-11 2022-05-03 浙江新和成股份有限公司 (S, S) -2, 8-diazabicyclo [4.3.0] nonane intermediate and preparation method and application thereof
CN110981874A (en) * 2020-03-05 2020-04-10 北京四环生物制药有限公司 Preparation method of moxifloxacin hydrochloride
CN112409352B (en) * 2020-11-20 2022-05-24 华南理工大学 Moxifloxacin drug derivatives and preparation method and application thereof
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Also Published As

Publication number Publication date
JP4111431B2 (en) 2008-07-02
FI113771B (en) 2004-06-15
FI930049A0 (en) 1993-01-07
TW209865B (en) 1993-07-21
CA2086914A1 (en) 1993-07-11
CN1043142C (en) 1999-04-28
AU669502B2 (en) 1996-06-13
HU9300034D0 (en) 1993-04-28
FI104174B1 (en) 1999-11-30
FI104174B (en) 1999-11-30
HU219488B (en) 2001-04-28
SK285155B6 (en) 2006-07-07
CN1075499C (en) 2001-11-28
CN1212256A (en) 1999-03-31
JP2003048890A (en) 2003-02-21
JP2003026574A (en) 2003-01-29
CZ289076B6 (en) 2001-10-17
FI930049A (en) 1993-07-11
AU3105493A (en) 1993-07-15
SK2212000A3 (en) 2006-05-04
FI110943B (en) 2003-04-30
SK282971B6 (en) 2003-01-09
SK285223B6 (en) 2006-09-07
CN1074218A (en) 1993-07-14
SK396692A3 (en) 2002-09-10
NO301420B1 (en) 1997-10-27
HUT64065A (en) 1993-11-29
CN1061351C (en) 2001-01-31
PL174853B1 (en) 1998-09-30
CZ396692A3 (en) 1993-08-11
CA2086914C (en) 2005-03-15
KR100251886B1 (en) 2000-07-01
JPH05271229A (en) 1993-10-19
CN1192440A (en) 1998-09-09
MX9207604A (en) 1993-10-01
EP0550903A1 (en) 1993-07-14
FI990207A0 (en) 1999-02-03
PL297338A1 (en) 1993-09-06
NO924978D0 (en) 1992-12-22
FI20020059A (en) 2002-01-11
SK2232000A3 (en) 2006-05-04
NO924978L (en) 1993-07-12
FI990207A (en) 1999-02-03
NZ245640A (en) 1995-03-28
KR930016421A (en) 1993-08-26

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