NO147382C - ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, FLUORATED AMINO ACIDS - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, FLUORATED AMINO ACIDS

Info

Publication number: NO147382C
Authority: NO; Norway
Prior art keywords: fluorated; preparation; amino acids; therapeutic active; analogy procedure
Prior art date: 1977-06-01

Application number

NO781892A

Other languages

Norwegian (no)

Other versions

NO781892L (en

NO147382B (en

Inventor

Janos Kollonitsch

Arthur Allan Patchett

Stephen Marburg

Original Assignee

Merck & Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-06-01

Filing date

1978-05-31

Publication date

1983-03-30

1977-06-01 Priority claimed from US05/802,391 external-priority patent/US4325961A/en

1978-05-31 Application filed by Merck & Co Inc filed Critical Merck & Co Inc

1978-12-04 Publication of NO781892L publication Critical patent/NO781892L/en

1982-12-20 Publication of NO147382B publication Critical patent/NO147382B/en

1983-03-30 Publication of NO147382C publication Critical patent/NO147382C/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)

NO781892A 1977-06-01 1978-05-31 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, FLUORATED AMINO ACIDS NO147382C (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US80238977A	1977-06-01	1977-06-01
US05/802,391 US4325961A (en)	1977-06-01	1977-06-01	Fluorinated amino acids

Publications (3)

Publication Number	Publication Date
NO781892L NO781892L (en)	1978-12-04
NO147382B NO147382B (en)	1982-12-20
NO147382C true NO147382C (en)	1983-03-30

Family

ID=27122442

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO781892A NO147382C (en)	1977-06-01	1978-05-31	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, FLUORATED AMINO ACIDS

Country Status (26)

Country	Link
JP (1)	JPS5416423A (en)
AR (1)	AR223463A1 (en)
AT (1)	AT360509B (en)
AU (1)	AU518479B2 (en)
CA (1)	CA1120040A (en)
CH (1)	CH639639A5 (en)
DD (1)	DD138651A5 (en)
DE (1)	DE2824116A1 (en)
DK (1)	DK149841C (en)
ES (1)	ES470296A1 (en)
FI (1)	FI66840C (en)
FR (1)	FR2392958A1 (en)
GB (1)	GB1602525A (en)
GR (1)	GR64495B (en)
HK (1)	HK18184A (en)
HU (1)	HU181911B (en)
IE (1)	IE46983B1 (en)
IT (1)	IT1104709B (en)
LU (1)	LU79750A1 (en)
NL (1)	NL190485C (en)
NO (1)	NO147382C (en)
NZ (1)	NZ187377A (en)
PL (1)	PL115731B1 (en)
PT (1)	PT68102B (en)
SE (1)	SE7806440L (en)
YU (1)	YU129178A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA783273B (en) *	1977-07-11	1979-06-27	Merrell Toraude & Co	A-halomethyl amino acids
IL59481A0 (en) *	1977-07-11	1980-05-30	Merrell Toraude & Co	-halomethyl amino acids
CA1091661A (en) *	1977-07-11	1980-12-16	Philippe Bey	.alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS
US4315095A (en) *	1977-07-28	1982-02-09	Merrell Toraude Et Compagnie	α-Halomethyl derivatives of amino acids
DE2965364D1 (en) *	1978-07-24	1983-06-16	Merck & Co Inc	Alpha-difluoromethyl amino acids and pharmaceutical composition containing the same
IE49522B1 (en) *	1979-04-26	1985-10-16	Merrell Toraude & Co	Alpha-halomethylaminoacids
IL60591A (en) *	1979-07-26	1985-02-28	Merrell Toraude & Co	Alkenyl fluoromethyl ketimine magnesium halides and process for their preparation
ZA813018B (en) *	1980-05-09	1982-05-26	Merrell Toraude & Co	Fluoromethylated tyrosine methyl ester
ZA813953B (en) *	1980-06-16	1982-06-30	Merrell Dow Pharma	Method of inhibiting the growth of protozoa
US4421767A (en) *	1981-06-01	1983-12-20	Merrell Toraude Et Compagnie	Compounds and methods for treating depression
GB9325368D0 (en) *	1993-12-10	1994-02-16	Univ Bristol	Organic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3046300A (en) *	1960-10-21	1962-07-24	Merck & Co Inc	alpha-trifluoromethyloxyphenylalanines

1978
- 1978-05-25 GR GR56328A patent/GR64495B/en unknown
- 1978-05-25 NZ NZ187377A patent/NZ187377A/en unknown
- 1978-05-25 FR FR7815567A patent/FR2392958A1/en active Granted
- 1978-05-26 AR AR272336A patent/AR223463A1/en active
- 1978-05-26 FI FI781674A patent/FI66840C/en not_active IP Right Cessation
- 1978-05-29 CA CA000304318A patent/CA1120040A/en not_active Expired
- 1978-05-29 AU AU36586/78A patent/AU518479B2/en not_active Expired
- 1978-05-29 ES ES470296A patent/ES470296A1/en not_active Expired
- 1978-05-30 DD DD78205669A patent/DD138651A5/en unknown
- 1978-05-30 HU HU78ME2169A patent/HU181911B/en unknown
- 1978-05-30 PT PT68102A patent/PT68102B/en unknown
- 1978-05-30 AT AT393278A patent/AT360509B/en not_active IP Right Cessation
- 1978-05-30 IE IE1078/78A patent/IE46983B1/en unknown
- 1978-05-30 DK DK237978A patent/DK149841C/en not_active IP Right Cessation
- 1978-05-30 GB GB24330/78A patent/GB1602525A/en not_active Expired
- 1978-05-30 YU YU01291/78A patent/YU129178A/en unknown
- 1978-05-31 CH CH597978A patent/CH639639A5/en not_active IP Right Cessation
- 1978-05-31 PL PL1978207242A patent/PL115731B1/en unknown
- 1978-05-31 IT IT49637/78A patent/IT1104709B/en active
- 1978-05-31 NO NO781892A patent/NO147382C/en unknown
- 1978-06-01 DE DE19782824116 patent/DE2824116A1/en active Granted
- 1978-06-01 NL NLAANVRAGE7805981,A patent/NL190485C/en not_active IP Right Cessation
- 1978-06-01 LU LU79750A patent/LU79750A1/en unknown
- 1978-06-01 SE SE7806440A patent/SE7806440L/en unknown
- 1978-06-01 JP JP6501678A patent/JPS5416423A/en active Granted
1984
- 1984-03-01 HK HK181/84A patent/HK18184A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
IE46983B1 (en)	1983-11-16
AR223463A1 (en)	1981-08-31
HU181911B (en)	1983-11-28
HK18184A (en)	1984-03-09
IE781078L (en)	1978-12-01
IT7849637A0 (en)	1978-05-31
AU3658678A (en)	1979-12-06
PT68102B (en)	1982-06-08
PL207242A1 (en)	1979-04-23
LU79750A1 (en)	1979-02-02
IT1104709B (en)	1985-10-28
FI781674A (en)	1978-12-02
GR64495B (en)	1980-03-31
FI66840C (en)	1984-12-10
DE2824116C2 (en)	1989-04-27
CA1120040A (en)	1982-03-16
DK149841B (en)	1986-10-13
NL190485B (en)	1993-10-18
NL7805981A (en)	1978-12-05
DK149841C (en)	1987-04-21
PL115731B1 (en)	1981-04-30
YU129178A (en)	1983-01-21
GB1602525A (en)	1981-11-11
SE7806440L (en)	1978-12-02
NO781892L (en)	1978-12-04
AT360509B (en)	1981-01-12
NL190485C (en)	1994-03-16
FR2392958A1 (en)	1978-12-29
CH639639A5 (en)	1983-11-30
ATA393278A (en)	1980-06-15
JPS641474B2 (en)	1989-01-11
NO147382B (en)	1982-12-20
DD138651A5 (en)	1979-11-14
DK237978A (en)	1979-01-19
AU518479B2 (en)	1981-10-01
ES470296A1 (en)	1979-09-16
FR2392958B1 (en)	1980-10-24
NZ187377A (en)	1981-05-15
FI66840B (en)	1984-08-31
PT68102A (en)	1978-06-01
JPS5416423A (en)	1979-02-07
DE2824116A1 (en)	1978-12-14

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