NO170081C - ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLD DERIVATIVES WITH ACTIVITY ON COLLINERY SYSTEM - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLD DERIVATIVES WITH ACTIVITY ON COLLINERY SYSTEM

Info

Publication number: NO170081C
Authority: NO; Norway
Prior art keywords: tiazold; collinery; derivatives; activity; preparation
Prior art date: 1987-03-12

Application number

NO881093A

Other languages

Norwegian (no)

Other versions

NO170081B (en

NO881093D0 (en

NO881093L (en

Inventor

Kathleen Biziere

Dominique Olliero

Paul Worms

Original Assignee

Sanofi Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-03-12

Filing date

1988-03-11

Publication date

1992-09-09

1988-03-11 Application filed by Sanofi Sa filed Critical Sanofi Sa

1988-03-11 Publication of NO881093D0 publication Critical patent/NO881093D0/en

1988-09-13 Publication of NO881093L publication Critical patent/NO881093L/en

1992-06-01 Publication of NO170081B publication Critical patent/NO170081B/en

1992-09-09 Publication of NO170081C publication Critical patent/NO170081C/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/84—Naphthothiazoles

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Pyridine Compounds (AREA)

NO881093A 1987-03-12 1988-03-11 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLD DERIVATIVES WITH ACTIVITY ON COLLINERY SYSTEM NO170081C (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8703398A FR2612187B1 (en)	1987-03-12	1987-03-12	THIAZOLE DERIVATIVES ACTIVE IN THE CHOLINERGIC SYSTEM, THEIR PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME

Publications (4)

Publication Number	Publication Date
NO881093D0 NO881093D0 (en)	1988-03-11
NO881093L NO881093L (en)	1988-09-13
NO170081B NO170081B (en)	1992-06-01
NO170081C true NO170081C (en)	1992-09-09

Family

ID=9348897

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO881093A NO170081C (en)	1987-03-12	1988-03-11	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLD DERIVATIVES WITH ACTIVITY ON COLLINERY SYSTEM

Country Status (27)

Country	Link
EP (1)	EP0283390B1 (en)
JP (1)	JPS63243080A (en)
KR (1)	KR880011135A (en)
AR (1)	AR243515A1 (en)
AT (1)	ATE86249T1 (en)
AU (1)	AU612350B2 (en)
DD (1)	DD274028A5 (en)
DE (1)	DE3878708T2 (en)
DK (1)	DK170162B1 (en)
ES (1)	ES2053778T3 (en)
FI (1)	FI881152A (en)
FR (1)	FR2612187B1 (en)
HU (1)	HU198916B (en)
IE (1)	IE60173B1 (en)
IL (1)	IL85704A (en)
MA (1)	MA21207A1 (en)
MY (1)	MY103233A (en)
NO (1)	NO170081C (en)
NZ (1)	NZ223845A (en)
OA (1)	OA08871A (en)
PH (1)	PH25389A (en)
PL (1)	PL151889B1 (en)
PT (1)	PT86952B (en)
SU (1)	SU1604157A3 (en)
TN (1)	TNSN88020A1 (en)
YU (1)	YU49688A (en)
ZA (1)	ZA881764B (en)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS6440474A (en) *	1987-08-04	1989-02-10	Hisamitsu Pharmaceutical Co	Novel 2-substituted aminothiazole derivative
JPH0753666B2 (en) *	1987-09-14	1995-06-07	久光製薬株式会社	Anti-inflammatory agent consisting of substituted diphenylthiazole derivative
FR2656610B1 (en) *	1989-12-29	1992-05-07	Sanofi Sa	DERIVATIVES OF 2-AMINO PHENYL-4 THIAZOLE, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION.
WO1991018882A1 (en) *	1990-05-29	1991-12-12	Nippon Soda Co., Ltd.	N-substituted heterocyclic amidine derivative
WO1992021666A1 (en) *	1991-05-31	1992-12-10	Laboratoires Upsa	Angiotensin ii receptor antagonist thiazole devivatives
FR2677021B1 (en) *	1991-05-31	1993-10-01	Upsa Laboratoires	NOVEL THIAZOLE DERIVATIVES ANTAGONISTS OF ANGIOTENSIN II RECEPTORS; THEIR PREPARATION METHODS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
FR2692893B1 (en) *	1992-06-24	1994-09-02	Sanofi Elf	Branched alkylamino thiazole derivatives, processes for their preparation and pharmaceutical compositions containing them.
WO1994020476A1 (en) *	1993-03-02	1994-09-15	Fujisawa Pharmaceutical Co., Ltd.	Novel heterocyclic compound
FR2714059B1 (en) *	1993-12-21	1996-03-08	Sanofi Elf	Branched amino derivatives of thiazole, processes for their preparation and pharmaceutical compositions containing them.
FR2735777B1 (en) *	1995-06-21	1997-09-12	Sanofi Sa	4-PHENYLAMINOTHIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FR2754258B1 (en) *	1996-10-08	1998-12-31	Sanofi Sa	AMINOTHIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
GB9705428D0 (en) *	1997-03-15	1997-04-30	Knoll Ag	Therapeutic agents
WO1999065884A1 (en) *	1998-06-18	1999-12-23	Bristol-Myers Squibb Company	Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
DE60034783T2 (en)	1999-04-22	2008-01-31	H. Lundbeck A/S, Valby	SELECTIVE NPY (Y5) ANTAGONISTS
US6340683B1 (en)	1999-04-22	2002-01-22	Synaptic Pharmaceutical Corporation	Selective NPY (Y5) antagonists (triazines)
US6218408B1 (en)	1999-06-30	2001-04-17	Synaptic Pharmaceutical Corporation	Selective NPY (Y5) antagonists (bicyclics)
US6989379B1 (en)	1999-04-22	2006-01-24	H. Lundbick A/S	Selective NPY (Y5) antagonists
US6214853B1 (en)	1999-06-30	2001-04-10	Synaptic Pharmaceutical Corporation	Selective NPY (Y5) antagonists (bicyclics)
US6222040B1 (en)	1999-06-30	2001-04-24	Synaptic Pharmaceutical Corporation	Selective NPY (Y5) antagonists (tricyclics)
US6225330B1 (en)	1999-06-30	2001-05-01	Synaptic Pharmaceutical Corporation	Selective NPY (Y5) antagonists (tricyclics)
US7273880B2 (en)	1999-06-30	2007-09-25	H. Lunbeck A/S	Selective NPY (Y5) antagonists
AU2002314744A1 (en)	2001-04-17	2002-10-28	Sepracor, Inc.	Thiazole and other heterocyclic ligands and use thereof
US7485655B2 (en) *	2002-01-16	2009-02-03	University Of Virginia Patent Foundation	2-Aminothiazole allosteric enhancers of A1 adenosine receptors
DE10251513A1 (en) *	2002-11-04	2004-05-19	Basf Ag	Compounds with 5-membered heterocycle linked by amino- or phosphino-methyl to a benzene ring with an ortho-hydroxy, alkoxy, thiol or amino group, used as multidentate ligands in olefin polymerization catalysts
JP2007261945A (en) *	2004-04-07	2007-10-11	Taisho Pharmaceut Co Ltd	Thiazole derivative
WO2006130493A2 (en) *	2005-05-31	2006-12-07	Vertex Pharmaceuticals Incorporated	Heterocycles useful as modulators of ion channels
KR20110137941A (en) *	2010-06-18	2011-12-26	(주) 에빅스젠	Novel thiourea or urea derivative, preparation method thereof and pharmaceutical composition for preventing or treating AIDS containing the same as an active ingredient
RU2456284C1 (en) *	2011-04-12	2012-07-20	Федеральное государственное автономное образовательное учреждение высшего профессионального образования "Уральский федеральный университет имени первого Президента России Б.Н. Ельцина"	2-aminopropylmorpholino-5-aryl-6h-1,3,4-thiadiazines, dihydrobromides and 2-aminopropylmorpholino-4-arylthiazoles, hydrobromides showing antiaggregant action
CA2967316C (en) *	2014-11-10	2021-12-14	Forge Life Science, Llc	Anti-hcmv compositions and methods
CN115160207B (en) *	2022-04-21	2023-09-26	烟台大学	Benzoyl thiourea compound, preparation method thereof and application of red tide algae algicide

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2975182A (en) *	1959-11-16	1961-03-14	Paul A J Janssen	1-(aroylalkyl)-4-(heterocyclyl) piperazines
FR2092714B1 (en) *	1970-06-11	1974-03-22	Melle Bezons
CH583232A5 (en) *	1973-02-02	1976-12-31	Wander Ag Dr A
DE3135250A1 (en) *	1981-09-05	1983-03-17	Basf Ag, 6700 Ludwigshafen	TRICYCLIC THIAZOLYLOXAMATES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM
US4552886A (en) *	1982-06-07	1985-11-12	Eli Lilly And Company	Fungicidal pyridylmethyl-amines
FR2581063B1 (en) *	1985-04-30	1987-07-17	Chauvin Blache Lab	AMINO-2 THIAZOLES N-SUBSTITUTED, THEIR PREPARATION PROCESS AND THEIR APPLICATION IN THERAPEUTICS
HUT43600A (en) *	1985-06-22	1987-11-30	Sandoz Ag	Process for production of new thiazole derivatives and medical compound containing those

1987
- 1987-03-12 FR FR8703398A patent/FR2612187B1/en not_active Expired
1988
- 1988-03-03 AU AU12662/88A patent/AU612350B2/en not_active Ceased
- 1988-03-08 MA MA21448A patent/MA21207A1/en unknown
- 1988-03-08 DD DD88313502A patent/DD274028A5/en not_active IP Right Cessation
- 1988-03-09 PH PH36616A patent/PH25389A/en unknown
- 1988-03-09 DK DK128688A patent/DK170162B1/en not_active IP Right Cessation
- 1988-03-10 NZ NZ223845A patent/NZ223845A/en unknown
- 1988-03-10 AR AR88310267A patent/AR243515A1/en active
- 1988-03-11 SU SU884355377A patent/SU1604157A3/en active
- 1988-03-11 ES ES88400572T patent/ES2053778T3/en not_active Expired - Lifetime
- 1988-03-11 NO NO881093A patent/NO170081C/en unknown
- 1988-03-11 OA OA59299A patent/OA08871A/en unknown
- 1988-03-11 FI FI881152A patent/FI881152A/en not_active Application Discontinuation
- 1988-03-11 ZA ZA881764A patent/ZA881764B/en unknown
- 1988-03-11 PT PT86952A patent/PT86952B/en not_active IP Right Cessation
- 1988-03-11 MY MYPI88000258A patent/MY103233A/en unknown
- 1988-03-11 YU YU00496/88A patent/YU49688A/en unknown
- 1988-03-11 EP EP88400572A patent/EP0283390B1/en not_active Expired - Lifetime
- 1988-03-11 DE DE8888400572T patent/DE3878708T2/en not_active Expired - Fee Related
- 1988-03-11 HU HU881190A patent/HU198916B/en not_active IP Right Cessation
- 1988-03-11 PL PL1988271132A patent/PL151889B1/en unknown
- 1988-03-11 IL IL85704A patent/IL85704A/en unknown
- 1988-03-11 AT AT88400572T patent/ATE86249T1/en not_active IP Right Cessation
- 1988-03-11 TN TNTNSN88020A patent/TNSN88020A1/en unknown
- 1988-03-11 IE IE72188A patent/IE60173B1/en not_active IP Right Cessation
- 1988-03-12 KR KR1019880002614A patent/KR880011135A/en not_active Application Discontinuation
- 1988-03-12 JP JP63059223A patent/JPS63243080A/en active Pending

Also Published As

Publication number	Publication date
ES2053778T3 (en)	1994-08-01
FR2612187A1 (en)	1988-09-16
HU198916B (en)	1989-12-28
MA21207A1 (en)	1988-10-01
KR880011135A (en)	1988-10-26
NO170081B (en)	1992-06-01
IE880721L (en)	1988-09-12
NZ223845A (en)	1990-11-27
DK170162B1 (en)	1995-06-06
AU612350B2 (en)	1991-07-11
PT86952A (en)	1988-04-01
ZA881764B (en)	1988-08-31
IL85704A (en)	1992-11-15
PL151889B1 (en)	1990-10-31
ATE86249T1 (en)	1993-03-15
FI881152A0 (en)	1988-03-11
DK128688A (en)	1988-09-13
PT86952B (en)	1992-05-29
PL271132A1 (en)	1988-11-24
MY103233A (en)	1993-05-29
YU49688A (en)	1989-10-31
IL85704A0 (en)	1988-08-31
AR243515A1 (en)	1993-08-31
OA08871A (en)	1989-10-31
DE3878708D1 (en)	1993-04-08
JPS63243080A (en)	1988-10-07
FI881152A (en)	1988-09-13
SU1604157A3 (en)	1990-10-30
EP0283390A3 (en)	1988-09-28
TNSN88020A1 (en)	1990-07-10
HUT47261A (en)	1989-02-28
NO881093D0 (en)	1988-03-11
FR2612187B1 (en)	1989-07-21
NO881093L (en)	1988-09-13
AU1266288A (en)	1988-09-15
IE60173B1 (en)	1994-06-15
DE3878708T2 (en)	1993-09-02
PH25389A (en)	1991-06-03
EP0283390A2 (en)	1988-09-21
DD274028A5 (en)	1989-12-06
DK128688D0 (en)	1988-03-09
EP0283390B1 (en)	1993-03-03

Publication	Publication Date	Title
NO170081C (en)	1992-09-09	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLD DERIVATIVES WITH ACTIVITY ON COLLINERY SYSTEM
NO883974D0 (en)	1988-09-07	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TETRAHYDRO-HYDROXYPYRANON DERIVATIVES.
NO864126D0 (en)	1986-10-16	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRIDON DERIVATIVES.
NO163406C (en)	1990-05-23	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOKINOLINO DERIVATIVES.
NO862477D0 (en)	1986-06-20	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-ARYLIMIDAZOLE DERIVATIVES.
NO853293L (en)	1986-02-24	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC DERIVATIVES.
NO171638C (en)	1993-04-14	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE QUINOLINE DERIVATIVES
NO884231D0 (en)	1988-09-23	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOPYRIDINE DERIVATIVES.
NO853100L (en)	1986-02-10	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZO PYRIDINES.
NO862956L (en)	1987-01-26	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRIMIDINE DERIVATIVES.
NO176275C (en)	1995-03-08	Analogous Process for the Preparation of Therapeutically Active Pyridazinone Derivatives
NO168355C (en)	1992-02-12	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZIMIDAZOLD DERIVATIVES
NO854369L (en)	1986-05-05	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZIMIDAZOLE DERIVATIVES
NO164897C (en)	1990-11-28	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE OXAZOLIDINON DERIVATIVES.
NO862372D0 (en)	1986-06-13	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE QUINOLO DERIVATIVES.
NO891114D0 (en)	1989-03-15	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ARAKIDONIC ACID DERIVATIVES.
NO884175L (en)	1989-03-22	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE HETEROCYCLIC DERIVATIVES.
NO167802C (en)	1991-12-11	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZOTIAZEPINE DERIVATIVES.
NO864101L (en)	1987-04-21	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DICHLORANILIN DERIVATIVES.
NO167668C (en)	1991-11-27	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE EPIPODOPHYLLOTOXING LUCOSIDE-4'-ACYL DERIVATIVES.
NO162072C (en)	1989-11-01	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TIENOPYRIDINE DERIVATIVES.
NO890607D0 (en)	1989-02-13	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRIDINE DERIVATIVES.
FI89595B (en)	1993-07-15	For the preparation of therapeutically active 2- (thioalkylamino) ethyl-1H-imidazole derivatives
NO165295C (en)	1991-01-30	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CEPHALOSPORIN DERIVATIVES.
NO852563L (en)	1985-12-30	PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRIDINE DERIVATIVES.