PT84770A - BENZOTHIAZINONE DERIVATIVES PROCESS FOR THEIR MANUFACTURE THEREOF AND THEIR USE - Google Patents

BENZOTHIAZINONE DERIVATIVES PROCESS FOR THEIR MANUFACTURE THEREOF AND THEIR USE

Info

Publication number
PT84770A
PT84770A PT84770A PT8477087A PT84770A PT 84770 A PT84770 A PT 84770A PT 84770 A PT84770 A PT 84770A PT 8477087 A PT8477087 A PT 8477087A PT 84770 A PT84770 A PT 84770A
Authority
PT
Portugal
Prior art keywords
manufacture
derivatives process
benzothiazinone derivatives
benzothiazinone
derivatives
Prior art date
Application number
PT84770A
Other languages
German (de)
Portuguese (pt)
Other versions
PT84770B (en
Inventor
Ulrich Lerch
Rainer Henning
Joachim Kaiser
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT84770A publication Critical patent/PT84770A/en
Publication of PT84770B publication Critical patent/PT84770B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/141,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/141,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/161,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT84770A 1986-04-28 1987-04-27 METHOD FOR PREPARING BENZOTIAZINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PT84770B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19863614363 DE3614363A1 (en) 1986-04-28 1986-04-28 BENZOTHIAZINONE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, MEDICINAL PRODUCTS CONTAINING THEM AND THE USE THEREOF

Publications (2)

Publication Number Publication Date
PT84770A true PT84770A (en) 1987-05-01
PT84770B PT84770B (en) 1989-12-29

Family

ID=6299713

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84770A PT84770B (en) 1986-04-28 1987-04-27 METHOD FOR PREPARING BENZOTIAZINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (13)

Country Link
EP (1) EP0244723A3 (en)
JP (1) JPS62258371A (en)
KR (1) KR870010028A (en)
AU (1) AU601659B2 (en)
DE (1) DE3614363A1 (en)
DK (1) DK213387A (en)
FI (1) FI871813A (en)
HU (1) HU199814B (en)
IL (1) IL82332A (en)
NO (1) NO871745L (en)
NZ (1) NZ220100A (en)
PT (1) PT84770B (en)
ZA (1) ZA872972B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3724366A1 (en) * 1987-07-23 1989-02-02 Hoechst Ag BENZOTHIAZINONE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, MEDICINAL PRODUCTS CONTAINING THEM AND THE USE THEREOF
DE3726759A1 (en) * 1987-08-12 1989-03-09 Hoechst Ag BENZOTHIAZINONE OXIDES, METHOD FOR THE PRODUCTION THEREOF, MEDICINAL PRODUCTS CONTAINING IT AND THEIR USE, AND INTERMEDIATE PRODUCTS FOR THEIR PRODUCTION
US5182276A (en) * 1989-06-16 1993-01-26 Santen Pharmaceutical Co., Ltd. Nootropic agent
US6207665B1 (en) 1997-06-12 2001-03-27 Schering Aktiengesellschaft Piperazine derivatives and their use as anti-inflammatory agents
US6693099B2 (en) * 2000-10-17 2004-02-17 The Procter & Gamble Company Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
BRPI0404222A (en) * 2004-06-07 2006-02-07 Fundacao Oswaldo Cruz Lidocaine derivatives, pharmaceutical compositions containing them, use of the respective pharmaceutical compositions in the treatment, prevention or inhibition of diseases as well as the method of treating, preventing or inhibiting diseases with said pharmaceutical compositions
JP6836502B2 (en) * 2014-05-30 2021-03-03 スプハエラ ファーマ ピーヴィーティー リミテッド New compound as an anti-tuberculosis drug

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59148771A (en) * 1983-02-09 1984-08-25 Santen Pharmaceut Co Ltd Benzothiazine derivative
US4584300A (en) * 1983-02-07 1986-04-22 Santen Pharmaceutical Co., Ltd. Platelet anti-aggregative- and calcium antagonistic -1,4-benzothiazin-3-one derivatives, compositions, and methods of use therefor
DE3347173A1 (en) * 1983-12-27 1985-07-04 Hoechst Ag, 6230 Frankfurt NEW BENZOTHIAZINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, MEDICINAL PRODUCTS CONTAINING THEM AND THE USE THEREOF
EP0186310A1 (en) * 1984-11-28 1986-07-02 Takeda Chemical Industries, Ltd. 1,4-Benzothiazine Derivatives, their production and use
EP0233291B1 (en) * 1985-03-19 1991-03-13 Santen Pharmaceutical Co., Ltd. 2-arylbenzothiazine derivatives
US4786635A (en) * 1985-07-29 1988-11-22 Santen Pharmaceutical Co., Ltd. Novel benzothiazine derivatives

Also Published As

Publication number Publication date
AU601659B2 (en) 1990-09-13
PT84770B (en) 1989-12-29
AU7199487A (en) 1987-10-29
FI871813A (en) 1987-10-29
DE3614363A1 (en) 1987-10-29
KR870010028A (en) 1987-11-30
JPS62258371A (en) 1987-11-10
DK213387A (en) 1987-10-29
NZ220100A (en) 1990-03-27
ZA872972B (en) 1987-11-25
DK213387D0 (en) 1987-04-27
EP0244723A2 (en) 1987-11-11
NO871745L (en) 1987-10-29
NO871745D0 (en) 1987-04-27
HUT45517A (en) 1988-07-28
HU199814B (en) 1990-03-28
IL82332A (en) 1991-08-16
EP0244723A3 (en) 1988-10-19
IL82332A0 (en) 1987-10-30
FI871813A0 (en) 1987-04-24

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MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19921231