UY30897A1 - Derivados de pentafluorotiobenzamidoacetonitrilo, composiciones conteniéndolos y aplicaciones - Google Patents

Derivados de pentafluorotiobenzamidoacetonitrilo, composiciones conteniéndolos y aplicaciones

Info

Publication number
UY30897A1
UY30897A1 UY30897A UY30897A UY30897A1 UY 30897 A1 UY30897 A1 UY 30897A1 UY 30897 A UY30897 A UY 30897A UY 30897 A UY30897 A UY 30897A UY 30897 A1 UY30897 A1 UY 30897A1
Authority
UY
Uruguay
Prior art keywords
compositions containing
pentafluorotiobenzamidoacetonitrile
derivatives
applications
compounds
Prior art date
Application number
UY30897A
Other languages
English (en)
Inventor
Yogest Anil Sabnis
Christelle Lauret
William Howson
Joanne Clare Hannam
Stuart Nicholas Complay
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of UY30897A1 publication Critical patent/UY30897A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/12—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom not containing sulfur-to-oxygen bonds, e.g. polysulfides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)

Abstract

La presente invencion se refiere a compuestos de formula (I) o un tautomero o profármaco de los mismos, o una sal farmacéuticamente aceptable de dicho compuesto, tautomero o profármaco, en la que: R1, R2, R3, R4, y R5 se selecciona cada uno independientemente de H, halogeno, CN, CF3 y CONH2; a composiciones que contienen dichos compuestos y a los usos de dichos compuestos como agentes antiparasitarios.
UY30897A 2007-02-09 2008-02-07 Derivados de pentafluorotiobenzamidoacetonitrilo, composiciones conteniéndolos y aplicaciones UY30897A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88904107P 2007-02-09 2007-02-09
US94682007P 2007-06-28 2007-06-28

Publications (1)

Publication Number Publication Date
UY30897A1 true UY30897A1 (es) 2008-09-30

Family

ID=39402647

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30897A UY30897A1 (es) 2007-02-09 2008-02-07 Derivados de pentafluorotiobenzamidoacetonitrilo, composiciones conteniéndolos y aplicaciones

Country Status (22)

Country Link
US (2) US7608604B2 (es)
EP (1) EP2118055B1 (es)
JP (1) JP4592819B2 (es)
KR (2) KR20110098012A (es)
AR (1) AR065280A1 (es)
AU (1) AU2008212594C1 (es)
BR (1) BRPI0807137A2 (es)
CA (1) CA2676147C (es)
CL (1) CL2008000403A1 (es)
CO (1) CO6220853A2 (es)
CY (1) CY1114932T1 (es)
DK (1) DK2118055T3 (es)
ES (1) ES2435191T3 (es)
HK (1) HK1133871A1 (es)
MX (1) MX2009007482A (es)
NZ (1) NZ578259A (es)
PL (1) PL2118055T3 (es)
PT (1) PT2118055E (es)
RU (1) RU2425825C2 (es)
TW (1) TWI352695B (es)
UY (1) UY30897A1 (es)
WO (1) WO2008096231A1 (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1380209E (pt) * 2001-04-17 2012-09-27 Nihon Nohyaku Co Ltd Composição de agente de controlo de pragas e método de utilização da mesma
DK2166855T3 (en) 2007-06-07 2018-06-14 Bayer Animal Health Gmbh COMBATING Ectoparasites
MX2010001133A (es) * 2007-07-30 2010-03-01 Du Pont Metodo de control de pulgas.
EA026649B1 (ru) 2008-10-21 2017-05-31 Мериал, Инк. Тиоамидные соединения, способ их получения и способ их применения
ES2551130T3 (es) 2008-11-14 2015-11-16 Merial, Inc. Compuestos de arilazol-2-ilcianoetilamino parasiticidas enriquecidos enantioméricamente
NZ592367A (en) 2008-12-03 2013-05-31 Novartis Ag Amidoacetonitrile compounds and pesticidal composition thereof
GB0905365D0 (en) 2009-03-27 2009-05-13 Norbrook Lab Ltd A topical parasiticide composition
TWI510189B (zh) 2009-06-19 2015-12-01 Lilly Co Eli 殺外寄生蟲之方法及調配物
EP2314292A1 (en) * 2009-10-20 2011-04-27 Novartis AG Endoparasiticidal compositions
KR20120098930A (ko) 2010-01-25 2012-09-05 일라이 릴리 앤드 캄파니 말과 말파리 유충을 내부적으로 억제 또는 처리하기 위한 방법
TWI580442B (zh) * 2011-10-19 2017-05-01 傑特大學 醫藥毫微懸浮物
JP2014530849A (ja) * 2011-10-19 2014-11-20 ゾエティス・エルエルシー 内部寄生虫に対するアミノアセトニトリル誘導体の使用
WO2013084860A1 (ja) * 2011-12-06 2013-06-13 宇部興産株式会社 ペンタフルオロスルファニル安息香酸の製造方法
RU2651761C2 (ru) * 2011-12-21 2018-04-23 Байер Интеллектуэль Проперти Гмбх Композиции, содержащие аморфный эмодепсид
CA2863384C (en) 2012-02-14 2017-08-29 Nippon Soda Co., Ltd. Aryloxyacetamide compound and pesticide
AU2013345149B2 (en) 2012-11-14 2016-10-27 Elanco Us Inc. Ectoparasiticidal methods and formulations
WO2014146750A1 (de) 2013-03-22 2014-09-25 Merck Patent Gmbh Synthesebausteine für die herstellung von materialien für organische elektrolumineszenzvorrichtungen
CN104230743B (zh) * 2013-06-24 2017-02-08 海正药业南通有限公司 一种4-苄基-1-苯乙基哌嗪-2,6-二酮的制备方法
AU2014286221B2 (en) * 2013-07-01 2018-05-31 The University Of Melbourne N-(1-cyano-2-hydroxy-1-methyl-ethyl)-4-(trifluoromethylsulfanyl)benzamide derivatives for use as nematocidal drugs
WO2016127350A1 (zh) 2015-02-12 2016-08-18 浙江海正药业股份有限公司 一种吡喹酮的制备方法及其中间体化合物
CN106018571A (zh) * 2015-11-09 2016-10-12 中华人民共和国淮安出入境检验检疫局 检测水生蔬菜中氯虫苯甲酰胺残留量的方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1643766A1 (de) * 1967-01-06 1971-07-01 Allied Chem Perhalogenierte Jodide sowie Verfahren zu ihrer Herstellung
GB9801851D0 (en) * 1998-01-29 1998-03-25 Pfizer Ltd Parasiticidal agents
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
EP1392281B1 (en) * 2000-12-20 2007-02-21 Novartis AG Anti-endoparasitic amidoacetonitrils
WO2002050052A1 (en) 2000-12-20 2002-06-27 Syngenta Participations Ag N-acyl aminoacetonitriles having pesticidal properties
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
DE10222192A1 (de) * 2002-05-18 2003-11-27 Aventis Pharma Gmbh Pentafluorsulfuranyl-benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10353205A1 (de) * 2003-11-13 2005-06-16 Aventis Pharma Deutschland Gmbh Ortho-substituierte Pentafluorsulfuranyl-Benzole, Verfahren zu ihrer Herstellung sowie ihre Verwendung als wertvolle Synthese-Zwischenstufen
US7514464B2 (en) * 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
US7425580B2 (en) 2004-05-19 2008-09-16 Wyeth (Diaryl-methyl)-malononitriles and their use as estrogen receptor ligands
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
EP1878249B1 (en) 2005-04-01 2020-03-04 LG Electronics, Inc. Method for scalably decoding a video signal

Also Published As

Publication number Publication date
KR20110098012A (ko) 2011-08-31
AU2008212594B2 (en) 2012-10-04
AU2008212594C1 (en) 2013-04-11
EP2118055A1 (en) 2009-11-18
CL2008000403A1 (es) 2008-08-18
PT2118055E (pt) 2013-11-19
CA2676147C (en) 2012-03-13
ES2435191T3 (es) 2013-12-16
US7608604B2 (en) 2009-10-27
JP2010518067A (ja) 2010-05-27
KR101136251B1 (ko) 2012-04-25
WO2008096231A1 (en) 2008-08-14
EP2118055B1 (en) 2013-08-21
BRPI0807137A2 (pt) 2014-04-15
TW200843728A (en) 2008-11-16
US20100010093A1 (en) 2010-01-14
RU2425825C2 (ru) 2011-08-10
CA2676147A1 (en) 2008-08-14
RU2009127356A (ru) 2011-03-20
NZ578259A (en) 2011-12-22
TWI352695B (en) 2011-11-21
HK1133871A1 (en) 2010-04-09
CO6220853A2 (es) 2010-11-19
AR065280A1 (es) 2009-05-27
US20080194694A1 (en) 2008-08-14
MX2009007482A (es) 2009-08-13
KR20090104856A (ko) 2009-10-06
DK2118055T3 (da) 2013-11-04
CY1114932T1 (el) 2016-12-14
WO2008096231A8 (en) 2009-08-20
JP4592819B2 (ja) 2010-12-08
AU2008212594A1 (en) 2008-08-14
PL2118055T3 (pl) 2014-01-31

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170908