DK158664C - METHOD OF ANALOGUE FOR THE PREPARATION OF BENZOXAZINONES AND BENZOXAZOLINONES AND RELATIONS FOR USING THE PROCEDURE. - Google Patents

METHOD OF ANALOGUE FOR THE PREPARATION OF BENZOXAZINONES AND BENZOXAZOLINONES AND RELATIONS FOR USING THE PROCEDURE.

Info

Publication number
DK158664C
DK158664C DK389082A DK389082A DK158664C DK 158664 C DK158664 C DK 158664C DK 389082 A DK389082 A DK 389082A DK 389082 A DK389082 A DK 389082A DK 158664 C DK158664 C DK 158664C
Authority
DK
Denmark
Prior art keywords
benzoxazolinones
benzoxazinones
relations
analogue
procedure
Prior art date
Application number
DK389082A
Other languages
Danish (da)
Other versions
DK389082A (en
DK158664B (en
Inventor
Kurt Schromm
Anton Mentrup
Ernst-Otto Renth
Armin Fuegner
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of DK389082A publication Critical patent/DK389082A/en
Publication of DK158664B publication Critical patent/DK158664B/en
Application granted granted Critical
Publication of DK158664C publication Critical patent/DK158664C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/341,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/361,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Feed For Specific Animals (AREA)
  • Fodder In General (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK389082A 1981-09-01 1982-08-31 METHOD OF ANALOGUE FOR THE PREPARATION OF BENZOXAZINONES AND BENZOXAZOLINONES AND RELATIONS FOR USING THE PROCEDURE. DK158664C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3134590 1981-09-01
DE19813134590 DE3134590A1 (en) 1981-09-01 1981-09-01 NEW BENZO HETEROCYCLES

Publications (3)

Publication Number Publication Date
DK389082A DK389082A (en) 1983-03-02
DK158664B DK158664B (en) 1990-07-02
DK158664C true DK158664C (en) 1991-01-14

Family

ID=6140603

Family Applications (1)

Application Number Title Priority Date Filing Date
DK389082A DK158664C (en) 1981-09-01 1982-08-31 METHOD OF ANALOGUE FOR THE PREPARATION OF BENZOXAZINONES AND BENZOXAZOLINONES AND RELATIONS FOR USING THE PROCEDURE.

Country Status (25)

Country Link
EP (1) EP0073505B1 (en)
JP (1) JPS5852278A (en)
KR (1) KR890000380B1 (en)
AR (2) AR231976A1 (en)
AT (1) ATE16703T1 (en)
AU (1) AU553589B2 (en)
CA (1) CA1180012A (en)
CS (1) CS236679B2 (en)
DD (1) DD204477A5 (en)
DE (2) DE3134590A1 (en)
DK (1) DK158664C (en)
ES (3) ES8308318A1 (en)
FI (1) FI78475C (en)
GB (1) GB2106105B (en)
GR (1) GR77275B (en)
HU (1) HU186112B (en)
IE (1) IE53615B1 (en)
IL (1) IL66683A0 (en)
NO (1) NO157738C (en)
NZ (1) NZ201777A (en)
PL (1) PL139375B1 (en)
PT (1) PT75478A (en)
SU (1) SU1149876A3 (en)
YU (1) YU42794B (en)
ZA (1) ZA826349B (en)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
DE3743265A1 (en) * 1987-12-19 1989-06-29 Boehringer Ingelheim Kg NEW AMMONIUM COMPOUNDS, THEIR MANUFACTURE AND USE
TW372967B (en) * 1994-12-27 1999-11-01 Kanebo Ltd 1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof
US7056916B2 (en) 2002-11-15 2006-06-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments for the treatment of chronic obstructive pulmonary disease
DE10253282A1 (en) 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Treatment of chronic obstructive pulmonary disease, using new or known N-substituted 2-amino-1-(benz-(1,4)-oxazin-3-on-8-yl)-ethanol derivative beta-mimetic agents, suitable for once-daily administration
PE20040950A1 (en) 2003-02-14 2005-01-01 Theravance Inc BIPHENYL DERIVATIVES AS AGONISTS OF ß2-ADRENERGIC RECEPTORS AND AS ANTAGONISTS OF MUSCARINAL RECEPTORS
BRPI0409198A (en) * 2003-04-04 2006-05-02 Novartis Ag quinolin-2-one derivatives for the treatment of airway diseases
GB0307856D0 (en) * 2003-04-04 2003-05-14 Novartis Ag Organic compounds
EP1789394A1 (en) * 2004-05-13 2007-05-30 Boehringer Ingelheim International Gmbh Hydroxy-substituted benzo-condensed heterocycles for use as beta agonists in the treatment of respiratory diseases
US7307076B2 (en) 2004-05-13 2007-12-11 Boehringer Ingelheim International Gmbh Beta agonists for the treatment of respiratory diseases
DE102004024454A1 (en) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Novel enantiomerically pure beta agonists, process for their preparation and their use as pharmaceuticals
DE102004024452A1 (en) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Aerosol formulation for the inhalation of beta agonists
US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
DE102004024451A1 (en) * 2004-05-14 2005-12-22 Boehringer Ingelheim Pharma Gmbh & Co. Kg Powder formulations for inhalation containing enantiomerically pure beta agonists
US7745621B2 (en) 2004-05-14 2010-06-29 Boehringer Ingelheim International Gmbh Long acting bronchodilators for the treatment of respiratory diseases
DE102004024453A1 (en) * 2004-05-14 2006-01-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg New long-acting bronchodilators for the treatment of respiratory diseases
JP5270343B2 (en) * 2005-08-15 2013-08-21 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Beta mimetic manufacturing method
TWI389692B (en) * 2005-10-10 2013-03-21 Boehringer Ingelheim Int Aerosol formulations for the inhalation of beta-agonists
GB0602778D0 (en) 2006-02-10 2006-03-22 Glaxo Group Ltd Novel compound
JP2010500319A (en) * 2006-08-07 2010-01-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Enantiomerically pure new beta agonists, methods for their preparation and their use as medicaments
UY30543A1 (en) * 2006-08-18 2008-03-31 Boehringer Ingelheim Int AEROSOL FORMULATION FOR INHALATION OF BETA- AGONISTS
TWI409071B (en) * 2007-01-25 2013-09-21 Boehringer Ingelheim Int Process for the manufacturing of beta mimentics

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035749A1 (en) * 1969-02-06 1970-12-24 Bellon Labor Sa Roger
CA1041523A (en) * 1974-06-19 1978-10-31 Queen's University Preparation of 1-oxapenicillins and novel intermediates therefor

Also Published As

Publication number Publication date
ES515380A0 (en) 1983-08-16
PL139375B1 (en) 1987-01-31
IE53615B1 (en) 1988-12-21
FI822985L (en) 1983-03-02
NO157738B (en) 1988-02-01
GB2106105A (en) 1983-04-07
ES8308318A1 (en) 1983-08-16
KR890000380B1 (en) 1989-03-15
CS236679B2 (en) 1985-05-15
JPH035392B2 (en) 1991-01-25
SU1149876A3 (en) 1985-04-07
AR231976A1 (en) 1985-04-30
ATE16703T1 (en) 1985-12-15
DE3134590A1 (en) 1983-03-10
YU42794B (en) 1988-12-31
FI78475C (en) 1989-08-10
YU194982A (en) 1984-12-31
IL66683A0 (en) 1982-12-31
EP0073505A1 (en) 1983-03-09
CA1180012A (en) 1984-12-27
NO157738C (en) 1988-05-11
IE822105L (en) 1983-03-01
HU186112B (en) 1985-06-28
AU8787482A (en) 1983-03-10
JPS5852278A (en) 1983-03-28
FI78475B (en) 1989-04-28
DK389082A (en) 1983-03-02
NZ201777A (en) 1985-08-30
NO822932L (en) 1983-03-02
DE3267702D1 (en) 1986-01-09
DD204477A5 (en) 1983-11-30
ES521871A0 (en) 1984-06-16
GB2106105B (en) 1985-07-10
DK158664B (en) 1990-07-02
ZA826349B (en) 1984-04-25
GR77275B (en) 1984-09-11
ES8402279A1 (en) 1984-01-16
ES521870A0 (en) 1984-01-16
EP0073505B1 (en) 1985-11-27
FI822985A0 (en) 1982-08-30
AU553589B2 (en) 1986-07-24
KR840001560A (en) 1984-05-07
AR231977A1 (en) 1985-04-30
PT75478A (en) 1982-09-01
ES8405778A1 (en) 1984-06-16
PL238077A1 (en) 1984-04-09

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