ES393554A1 - Thiazole derivatives and a process for the manufacture thereof - Google Patents

Thiazole derivatives and a process for the manufacture thereof

Info

Publication number
ES393554A1
ES393554A1 ES393554A ES393554A ES393554A1 ES 393554 A1 ES393554 A1 ES 393554A1 ES 393554 A ES393554 A ES 393554A ES 393554 A ES393554 A ES 393554A ES 393554 A1 ES393554 A1 ES 393554A1
Authority
ES
Spain
Prior art keywords
lower alkyl
formula
see formula
compound
thiazole derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES393554A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of ES393554A1 publication Critical patent/ES393554A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

A procedure for the preparation of thiazole derivatives of the formula ** (See formula) ** in which R1 represents a lower alkyl group and R2 represents lower aryl-lower alkyl or R1 and R2, together with the nitrogen atom to which they are attached, represent a hexagonal, heptagonal or octagonal pentagonal saturated heterocyclic ring, which may contain an oxygen atom and be replaced by one or more lower alkyl groups; and R3 represents a hydrogen atom or a lower alkyl group, and of the respective acid addition salts, characterized by: reacting a compound of the general formula ** (See formula) ** with a compound of the general formula ** (See formula) ** in which formulas the substituents have the meaning expressed above, and X represents a lower aryl group containing 6 to 12 carbon atoms. (Machine-translation by Google Translate, not legally binding)
ES393554A 1970-07-24 1971-07-23 Thiazole derivatives and a process for the manufacture thereof Expired ES393554A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1123970A CH543535A (en) 1970-07-24 1970-07-24 Process for the preparation of thiazole derivatives

Publications (1)

Publication Number Publication Date
ES393554A1 true ES393554A1 (en) 1974-11-16

Family

ID=4371497

Family Applications (1)

Application Number Title Priority Date Filing Date
ES393554A Expired ES393554A1 (en) 1970-07-24 1971-07-23 Thiazole derivatives and a process for the manufacture thereof

Country Status (15)

Country Link
AR (1) AR192413A1 (en)
AT (2) AT315168B (en)
AU (1) AU3041871A (en)
BE (1) BE770402A (en)
BR (1) BR7104636D0 (en)
CA (1) CA954514A (en)
CH (1) CH543535A (en)
DE (1) DE2137046A1 (en)
ES (1) ES393554A1 (en)
FR (2) FR2100949B1 (en)
GB (2) GB1355033A (en)
HU (1) HU163282B (en)
IL (1) IL37234A0 (en)
NL (1) NL7109995A (en)
ZA (1) ZA714030B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL102548A (en) * 1991-08-02 1998-08-16 Medivir Ab Thiourea derivatives for use in the preparation of medicaments for the inhibition of hiv and the treatment of aids and some such novel compounds
US5593993A (en) * 1991-08-02 1997-01-14 Medivir Ab Method for inhibition of HIV related viruses
CN108938628A (en) * 2018-08-29 2018-12-07 锁浩 A kind of composition and its application with anti-malarial activity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1265810A (en) * 1956-04-13 1961-07-07 Merck & Co Inc Process for the preparation of urea and thiourea derivatives
FR1533184A (en) * 1965-04-06 1968-07-19 Pechiney Saint Gobain Thiazole derivatives

Also Published As

Publication number Publication date
GB1355033A (en) 1974-06-05
GB1330930A (en) 1973-09-19
AT309420B (en) 1973-08-27
BE770402A (en) 1972-01-24
AR192413A1 (en) 1973-02-21
BR7104636D0 (en) 1973-03-08
FR2100949B1 (en) 1975-02-07
HU163282B (en) 1973-07-28
IL37234A0 (en) 1971-10-20
NL7109995A (en) 1972-01-26
CA954514A (en) 1974-09-10
FR2158578A1 (en) 1973-06-15
FR2100949A1 (en) 1972-03-24
CH543535A (en) 1973-10-31
FR2158578B1 (en) 1976-03-05
DE2137046A1 (en) 1972-01-27
AU3041871A (en) 1973-01-04
AT315168B (en) 1974-05-10
ZA714030B (en) 1972-03-29

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