IT1094209B - SEMI-SYNTHETIC ERITHROMYCIN DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION - Google Patents

SEMI-SYNTHETIC ERITHROMYCIN DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION

Info

Publication number
IT1094209B
IT1094209B IT20005/78A IT2000578A IT1094209B IT 1094209 B IT1094209 B IT 1094209B IT 20005/78 A IT20005/78 A IT 20005/78A IT 2000578 A IT2000578 A IT 2000578A IT 1094209 B IT1094209 B IT 1094209B
Authority
IT
Italy
Prior art keywords
erithromycin
derivatives
semi
synthetic
procedure
Prior art date
Application number
IT20005/78A
Other languages
Italian (it)
Other versions
IT7820005A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/856,479 external-priority patent/US4150220A/en
Application filed by Pfizer filed Critical Pfizer
Publication of IT7820005A0 publication Critical patent/IT7820005A0/en
Application granted granted Critical
Publication of IT1094209B publication Critical patent/IT1094209B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT20005/78A 1977-02-04 1978-02-03 SEMI-SYNTHETIC ERITHROMYCIN DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION IT1094209B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76548077A 1977-02-04 1977-02-04
US05/856,479 US4150220A (en) 1977-02-04 1977-12-01 Semi-synthetic 4"-erythromycin A derivatives

Publications (2)

Publication Number Publication Date
IT7820005A0 IT7820005A0 (en) 1978-02-03
IT1094209B true IT1094209B (en) 1985-07-26

Family

ID=27117613

Family Applications (1)

Application Number Title Priority Date Filing Date
IT20005/78A IT1094209B (en) 1977-02-04 1978-02-03 SEMI-SYNTHETIC ERITHROMYCIN DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION

Country Status (30)

Country Link
JP (1) JPS5827798B2 (en)
AR (1) AR222147A1 (en)
AU (1) AU501298B1 (en)
BG (2) BG32718A3 (en)
CA (1) CA1106367A (en)
CH (1) CH628906A5 (en)
CS (1) CS221801B2 (en)
DD (1) DD140048A5 (en)
DE (1) DE2804507C2 (en)
DK (1) DK148036C (en)
ES (2) ES466057A1 (en)
FI (1) FI780354A (en)
FR (2) FR2379550A1 (en)
GB (2) GB1585316A (en)
GR (1) GR68691B (en)
HU (1) HU182559B (en)
IE (1) IE46661B1 (en)
IL (2) IL53968A0 (en)
IT (1) IT1094209B (en)
LU (1) LU79004A1 (en)
NL (1) NL176174C (en)
NO (2) NO146472C (en)
NZ (1) NZ186385A (en)
PH (2) PH14421A (en)
PL (1) PL116228B1 (en)
PT (1) PT67568B (en)
RO (4) RO79686A7 (en)
SE (2) SE445223B (en)
SU (1) SU927122A3 (en)
YU (3) YU40913B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4382085A (en) * 1982-03-01 1983-05-03 Pfizer Inc. 4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
HN1998000074A (en) * 1997-06-11 1999-01-08 Pfizer Prod Inc DERIVATIVES FROM MACROLIDES C-4 SUBSTITUTED
US6407074B1 (en) 1997-06-11 2002-06-18 Pfizer Inc C-4″-substituted macrolide derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

Also Published As

Publication number Publication date
NL176174B (en) 1984-10-01
AU501298B1 (en) 1979-06-14
DD140048A5 (en) 1980-02-06
DE2804507A1 (en) 1978-08-10
NO150484B (en) 1984-07-16
NO811913L (en) 1978-08-07
PH16675A (en) 1983-12-13
SE445223B (en) 1986-06-09
DK148036B (en) 1985-02-11
NL7801262A (en) 1978-08-08
RO81622B (en) 1983-04-30
YU26583A (en) 1984-02-29
FR2385735A1 (en) 1978-10-27
FR2379550B1 (en) 1980-07-04
ES472429A1 (en) 1979-04-01
IT7820005A0 (en) 1978-02-03
BG33159A3 (en) 1982-12-15
ES466057A1 (en) 1978-10-01
SU927122A3 (en) 1982-05-07
CS221801B2 (en) 1983-04-29
PH14421A (en) 1981-07-10
YU40799B (en) 1986-06-30
GB1585315A (en) 1981-02-25
JPS5827798B2 (en) 1983-06-11
PL116228B1 (en) 1981-05-30
SE8300870D0 (en) 1983-02-16
IE780239L (en) 1978-08-04
IL53968A0 (en) 1978-04-30
NL176174C (en) 1985-03-01
NO146472B (en) 1982-06-28
YU7378A (en) 1983-04-30
HU182559B (en) 1984-02-28
GR68691B (en) 1982-02-01
NO146472C (en) 1982-10-06
DK51878A (en) 1978-08-05
DE2804507C2 (en) 1982-11-04
NO150484C (en) 1984-10-24
RO81622A (en) 1983-04-29
RO79686A7 (en) 1982-08-17
JPS53101337A (en) 1978-09-04
YU40913B (en) 1986-08-31
DK148036C (en) 1985-07-15
RO77345A (en) 1981-08-17
SE457086B (en) 1988-11-28
IL61997A0 (en) 1981-02-27
SE7800270L (en) 1978-08-05
BG32718A3 (en) 1982-09-15
AR222147A1 (en) 1981-04-30
CA1106367A (en) 1981-08-04
LU79004A1 (en) 1979-09-06
PT67568B (en) 1979-06-18
GB1585316A (en) 1981-02-25
YU227983A (en) 1984-04-30
FR2385735B1 (en) 1980-10-24
RO79687A7 (en) 1982-08-17
IE46661B1 (en) 1983-08-24
FI780354A (en) 1978-08-05
NO780389L (en) 1978-08-07
PT67568A (en) 1978-02-01
FR2379550A1 (en) 1978-09-01
YU40798B (en) 1986-06-30
NZ186385A (en) 1980-10-08
CH628906A5 (en) 1982-03-31
PL204428A1 (en) 1979-06-04
SE8300870L (en) 1983-02-16

Similar Documents

Publication Publication Date Title
IT1088554B (en) SELLECTIVE PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 7-INDROSSI CUMARINA
IT1098042B (en) MITROIMMIDAZOLI AND PROCEDURE FOR THEIR PREPARATION
IT1106176B (en) PIRROLO DERIVATIVES THEIR PREPARATION PROCEDURE AND THEIR THERAPEUTIC APPLICATION
IT1160264B (en) PROSTACYCLINE DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1158712B (en) ALCHILEN-AMMINE DERIVATIVE AND PROCEDURE FOR THEIR PREPARATION
IT1102755B (en) DERIVATIVES OF FEPTIDES AND THEIR PREPARATION
IT7849859A0 (en) 2-BENZOIL-4-CHLORO-GLYC DERIVATIVES SUBSTITUTED NANILIDS THEIR PREPARATION PROCEDURE AND THEIR THERAPEUTIC APPLICATION
IT1094314B (en) PROCEDURE FOR THE PREPARATION OF DIAZEPIN DERIVATIVES
IT1102816B (en) AMINO-ALCOXYFINYL DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1188970B (en) MORANOLINA DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1105454B (en) PROCEDURE FOR THE PREPARATION OF AMILORIDE AND ITS DERIVATIVES 6-REPLACED
IT1121483B (en) BENZOTIEPINIC DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1108968B (en) ACETYLENPROSTAGLANDINE AND PROCEDURE FOR THEIR PREPARATION
IT1156441B (en) PROCEDURE FOR THE PREPARATION OF FENYL AMMIDINE DERIVATIVES
IT1109400B (en) 2-AMINOMETHYL-PHENOL DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1147741B (en) EBURNANO HYDROXYMINE DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1132403B (en) ALOVINCAMONE DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT7825800A0 (en) PROCEDURE FOR THE MANUFACTURE OF P-HYDROXYPHENILGLYCINE AND ITS DERIVATIVES
IT1094209B (en) SEMI-SYNTHETIC ERITHROMYCIN DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1107653B (en) IMIDAZO-CHINOLIN-DIONI AND PROCEDURE FOR THEIR PREPARATION
IT7819332A0 (en) SULFONYDRAZONE DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION.
IT1160661B (en) PROSTACYCLIN INCLUSION COMPLEXES AND PROSTACYCLIN DERIVATIVES WITH CYCLODESTRINE AND PROCEDURE FOR THEIR PREPARATION
IT1106130B (en) 24-DEHYDROVITAMIN D3 DERIVATIVES AND THEIR PREPARATION
IT1132404B (en) 10-ALO-E-OMOEBURNANO DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1212412B (en) BENZO-AS-TRIAZINE DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION.